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- [31] Optimisation of a series of potent, selective and orally bioavailable GlyT1 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (08) : 2235 - 2239Thomson, Joanne L.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, EnglandBlackaby, Wesley P.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, EnglandJennings, Andrew S. R.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, EnglandGoodacre, Simon C.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, EnglandPike, Andrew论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, EnglandThomas, Steve论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, EnglandBrown, Terry A.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, EnglandSmith, Alison论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, EnglandPillai, Gopalan论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, EnglandStreet, Leslie J.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, EnglandLewis, Richard T.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England Merck Sharp & Dohme Ltd, Neurosci Res Ctr, Dept Med Chem, Harlow CM20 2QR, Essex, England
- [32] Discovery of potent and orally bioavailable 17β-hydroxysteroid dehydrogenase type 3 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY, 2012, 20 (10) : 3242 - 3254Harada, Koichiro论文数: 0 引用数: 0 h-index: 0机构: Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanKubo, Hideki论文数: 0 引用数: 0 h-index: 0机构: Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanAbe, Jun论文数: 0 引用数: 0 h-index: 0机构: Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanHaneta, Mari论文数: 0 引用数: 0 h-index: 0机构: Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanConception, Arnel论文数: 0 引用数: 0 h-index: 0机构: Sumika Technoserv Corp, Div Organ Synth, Takarazuka, Hyogo 6650051, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanInoue, Shinichi论文数: 0 引用数: 0 h-index: 0机构: Sumika Technoserv Corp, Div Organ Synth, Takarazuka, Hyogo 6650051, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanOkada, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Sumika Technoserv Corp, Div Organ Synth, Takarazuka, Hyogo 6650051, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, JapanNishioka, Kazuhiko论文数: 0 引用数: 0 h-index: 0机构: Sumitomo Chem Co Ltd, Crop Protect Div Int, Chuo Ku, Tokyo 1048260, Japan Sumitomo Chem Co Ltd, Environm Hlth Sci Lab, Konohana Ku, Osaka 5548558, Japan
- [33] Discovery of β-benzamido hydroxamic acids as potent, selective, and orally bioavailable TACE inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (01) : 241 - 246Duan, James J. -W.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAChen, Lihua论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USALu, Zhonghui论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAXue, Chu-Biao论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USALiu, Rui-Qin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USACovington, Maryanne B.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAQian, Mingxin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAWasserman, Zelda R.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAVaddi, Krishna论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USAChrist, David D.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USATrzaskos, James M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USANewton, Robert C.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USADecicco, Carl P.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Res & Dev, Princeton, NJ 08543 USA
- [34] Development of Novel Dual Binders as Potent, Selective, and Orally Bioavailable Tankyrase InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2013, 56 (24) : 10003 - 10015Hua, Zihao论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USABregman, Howard论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USABuchanan, John L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAChakka, Nagasree论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAGuzman-Perez, Angel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAGunaydin, Hakan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAHuang, Xin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAGu, Yan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USABerry, Virginia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USALiu, Jingzhou论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USATeffera, Yohannes论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAHuang, Liyue论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAEgge, Bryan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Bioassay & Profiling, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAEmkey, Renee论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Bioassay & Profiling, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAMullady, Erin L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Bioassay & Profiling, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USASchneider, Steve论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Bioassay & Profiling, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAAndrews, Paul S.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Bioassay & Profiling, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAAcquaviva, Lisa论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USADovey, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAMishra, Ankita论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USANewcomb, John论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USASaffran, Douglas论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USASerafino, Randy论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAStrathdee, Craig A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USATurci, Susan M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAStanton, Mary论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmaceut, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USAWilson, Cindy论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USADiMauro, Erin F.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Chem Res & Discovery, Cambridge, MA 02142 USA
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