Efficient, mild synthesis of N-unsubstituted 1,2,3-triazoles from methanolysis of 1-sulfonyl-1,2,3-triazoles

被引：6

作者：

Rodriguez-Florencio, Janeth ^{[1
]}

Martinez-Otero, Diego ^{[1
]}

Garcia-Eleno, Marco A. ^{[1
]}

Cuevas-Yanez, Erick ^{[1
]}

机构：

[1] Ctr Conjunto Invest Quim Sustentable UAEM UNAM, Toluca, Estado De Mexic, Mexico

来源：

SYNTHETIC COMMUNICATIONS | 2018年 / 48卷 / 17期

关键词：

N-Unsubstituted 1,2,3-triazoles; methanolysis; 1-sulfonyl-1,2,3-triazoles; ONE-POT SYNTHESIS; SULFONYL; CYCLOADDITION; ALKYNE; AZIDE; 4-ARYL-1H-1,2,3-TRIAZOLES; 1H-1,2,3-TRIAZOLES; NH-1,2,3-TRIAZOLES; DEPROTECTION; MAGNESIUM;

D O I：

10.1080/00397911.2018.1484485

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A small library of diverse N-unsubstituted 1,2,3-triazoles was prepared from the corresponding 1-sulfonyl-1,2,3-triazoles, which were treated only with MeOH at reflux temperature. This process was carried out in good yields showing high efficiency and good functional group tolerance. [GRAPHICS] .

引用

页码：2189 / 2197

页数：9

共 50 条

[41] Recent Applications of Click Reaction in the Syntheses of 1,2,3-triazoles
Heravi, Majid M.
Hamidi, Hoda
Zadsirjan, Vahideh
CURRENT ORGANIC SYNTHESIS, 2014, 11 (05) : 647 - 675
[42] Sulfonyl-1,2,3-Triazoles: Convenient Synthones for Heterocyclic Compounds
Zibinsky, Mikhail
Fokin, Valery V.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2013, 52 (05) : 1507 - 1510
[43] The impact of 1,2,3-triazoles in the design of functional coatings
Kantheti, Sasidhar
Narayan, Ramanuj
Raju, K. V. S. N.
RSC ADVANCES, 2015, 5 (05) : 3687 - 3708
[44] Medicinal attributes of 1,2,3-triazoles: Current developments
Dheer, Divya
Singh, Virender
Shankar, Ravi
BIOORGANIC CHEMISTRY, 2017, 71 : 30 - 54
[45] 1,2,3-Triazoles: general and key synthetic strategies
Santos, Cosme Silva
de Oliveira, Romario Jonas
de Oliveira, Ronaldo Nascimento
Rufino Freitas, Juliano Carlo
ARKIVOC, 2020, : 219 - 271
[46] Developments in the Application of 1,2,3-Triazoles in Cancer Treatment
Slavova, Katerina, I
Todorov, Lozan T.
Belskaya, Nataliya P.
Alcolea Palafox, Mauricio
Kostova, Irena P.
RECENT PATENTS ON ANTI-CANCER DRUG DISCOVERY, 2020, 15 (02) : 92 - 112
[47] A Concise Account of Synthetic Approaches to 1,2,3-Triazoles
Shaikh, Mubarak H.
Nagargoje, Amol A.
Tamboli, Yasinalli
Islam, Imadul
Shingate, Bapurao B.
ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL, 2024, 56 (06) : 523 - 555
[48] One-pot synthesis of 1,2,3-triazoles from Michael reaction
Korea Research Institute of Chemical Technology, Daejeon 305-343, Korea, Republic of
不详
Bull. Korean Chem. Soc., 2008, 4 (723-724): : 723 - 724
[49] Efficient one-pot synthesis of 1,2,3-triazoles from benzyl and alkyl halides
Kacprzak, K
SYNLETT, 2005, (06) : 943 - 946
[50] One-pot synthesis of 1,2,3-triazoles from Michael reaction
Lee, Ihl Young Choi
Yu, Ok Jong
Lim, Hee-Jeong
Lee, Hyo Won
BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2008, 29 (04): : 723 - 724

← 1 2 3 4 5 →