Efficient, mild synthesis of N-unsubstituted 1,2,3-triazoles from methanolysis of 1-sulfonyl-1,2,3-triazoles

被引：6

作者：

Rodriguez-Florencio, Janeth ^{[1
]}

Martinez-Otero, Diego ^{[1
]}

Garcia-Eleno, Marco A. ^{[1
]}

Cuevas-Yanez, Erick ^{[1
]}

机构：

[1] Ctr Conjunto Invest Quim Sustentable UAEM UNAM, Toluca, Estado De Mexic, Mexico

来源：

SYNTHETIC COMMUNICATIONS | 2018年 / 48卷 / 17期

关键词：

N-Unsubstituted 1,2,3-triazoles; methanolysis; 1-sulfonyl-1,2,3-triazoles; ONE-POT SYNTHESIS; SULFONYL; CYCLOADDITION; ALKYNE; AZIDE; 4-ARYL-1H-1,2,3-TRIAZOLES; 1H-1,2,3-TRIAZOLES; NH-1,2,3-TRIAZOLES; DEPROTECTION; MAGNESIUM;

D O I：

10.1080/00397911.2018.1484485

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A small library of diverse N-unsubstituted 1,2,3-triazoles was prepared from the corresponding 1-sulfonyl-1,2,3-triazoles, which were treated only with MeOH at reflux temperature. This process was carried out in good yields showing high efficiency and good functional group tolerance. [GRAPHICS] .

引用

页码：2189 / 2197

页数：9

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