Reaction of (E)-3-(Benzo[d][1,3]dioxol-5-yl)-2-Cyanoacryloyl Chloride with Nucleophilic Reagents Containing Nitrogen and Sulfur

被引：4
作者：
Shiba, S. A. [1 ]
El-Ziaty, A. K. [1 ]
El-Aasar, N. K. [1 ]
Al-Saman, H. A. [1 ]
机构：
[1] Ain Shams Univ, Fac Sci, Dept Chem, Cairo, Egypt
来源：
PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS | 2010年 / 185卷 / 08期
关键词：
Benzimidazoles; benzothiazipines; 2-cyanoacryloyl chloride; pyrimidinethiones; QUANTUM FORCE-FIELD; DERIVATIVES; ACID; THIAZEPINES; INHIBITION; OXAZEPINES;
D O I：
10.1080/10426500903176547
中图分类号：
O61 [无机化学];
学科分类号：
070301 ; 081704 ;
摘要：
(E)-3-(Benzo[d][1,3]dioxol-5-yl)-2-cyanoacryloyl chloride was reacted with nucleophilic reagents containing nitrogen and sulfur to give new acryloyl amides, imides, thioesters, and heterocyclic systems. Some of these products showed moderate activities against antibacterial and antifungal agents. Supplemental materials are available for this article. Go to the publisher's online edition of Phosphorus, Sulfur, and Silicon and the Related Elements to view the free supplemental file.
引用
收藏
页码：1645 / 1657
页数：13
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