Rational design of small molecule inhibitors of the Myc-Max transcription factor dimerization interface

被引:0
|
作者
O'Brien, Jeremy [1 ]
Bonham, Andrew [1 ]
机构
[1] Metropolitan State Univ Denver, Dept Chem, Denver, CO 80204 USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
939-CHED
引用
收藏
页数:1
相关论文
共 50 条
  • [31] Rational Design of Small Molecule Inhibitors Targeting RhoA Subfamily Rho GTPases
    Shang, Xun
    Marchioni, Fillipo
    Sipes, Nisha
    Evelyn, Chris R.
    Jerabek-Willemsen, Moran
    Duhr, Stefan
    Seibel, William
    Wortman, Matthew
    Zheng, Yi
    CHEMISTRY & BIOLOGY, 2012, 19 (06): : 699 - 710
  • [32] Small molecule inhibitors targeting Myc in embryonal tumors
    Castelletti, Deborah
    Fiaschetti, Giulio
    Berg, Thorsten
    Alexandre, Arcaro
    Grotzer, Michael
    CANCER RESEARCH, 2009, 69
  • [33] Small molecule transcription factor mimic
    Kwonj, Y
    Arndt, HD
    Qian, M
    Choi, Y
    Kawazoe, Y
    Dervan, PB
    Uesugi, M
    JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2004, 126 (49) : 15940 - 15941
  • [34] X-ray structures of Myc-Max and Mad-Max recognizing DNA: Molecular bases of regulation by proto-oncogenic transcription factors
    Nair, SK
    Burley, SK
    CELL, 2003, 112 (02) : 193 - 205
  • [35] Design of peptidic inhibitors targeting the dimerization interface of galectins
    Gagnon, Jacinthe
    Egesborg, Philippe
    Vladoiu, Maria Claudia
    St-Pierre, Yves
    Chatenet, David
    Doucet, Olas
    ACTA CRYSTALLOGRAPHICA A-FOUNDATION AND ADVANCES, 2017, 73 : C99 - C99
  • [36] Small molecule selectively suppresses MYC transcription in cancer cells
    Bouvard, Claire
    Lim, Sang Min
    Ludka, John
    Yazdani, Nahid
    Woods, Ashley K.
    Chatterjee, Arnab K.
    Schultz, Peter G.
    Zhu, Shoutian
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2017, 114 (13) : 3497 - 3502
  • [37] Control of lymphocyte development by the the Mad/Max/Myc transcription factor network
    Iritani, BM
    Gomez, I
    Carlos, LS
    Eisenman, RN
    FASEB JOURNAL, 2000, 14 (06): : A1034 - A1034
  • [38] Rational Design of Small Molecule Immune Checkpoints' Inhibitors: The PD-1 Challenge
    Barakat, Khaled
    JOURNAL OF PHARMACY AND PHARMACEUTICAL SCIENCES, 2017, 20 : 9S - 10S
  • [39] Rational Design of Small Molecule Inhibitors Targeting the Ras GEF, SOS1
    Evelyn, Chris R.
    Duan, Xin
    Biesiada, Jacek
    Seibel, William L.
    Meller, Jaroslaw
    Zheng, Yi
    CHEMISTRY & BIOLOGY, 2014, 21 (12): : 1618 - 1628
  • [40] Rational Design and Identification of Small-Molecule Allosteric Inhibitors of CD38
    Yang, Lixin
    Li, Ting
    Li, Songlu
    Wu, Yang
    Shi, Xiaomeng
    Jin, Hongwei
    Liu, Zhenming
    Zhao, Yongjuan
    Zhang, Liangren
    Lee, Hon Cheung
    Zhang, Lihe
    CHEMBIOCHEM, 2019, 20 (19) : 2485 - 2493