共 27 条
MMP-2 responsive polymeric micelles for cancer-targeted intracellular drug delivery
被引:108
作者:

Chen, Wei-Hai
论文数: 0 引用数: 0
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机构: Wuhan Univ, Key Lab Biomed Polymers, Minist Educ, Wuhan 430072, Peoples R China

Luo, Guo-Feng
论文数: 0 引用数: 0
h-index: 0
机构: Wuhan Univ, Key Lab Biomed Polymers, Minist Educ, Wuhan 430072, Peoples R China

Lei, Qi
论文数: 0 引用数: 0
h-index: 0
机构: Wuhan Univ, Key Lab Biomed Polymers, Minist Educ, Wuhan 430072, Peoples R China

Jia, Hui-Zhen
论文数: 0 引用数: 0
h-index: 0
机构: Wuhan Univ, Key Lab Biomed Polymers, Minist Educ, Wuhan 430072, Peoples R China

Hong, Sheng
论文数: 0 引用数: 0
h-index: 0
机构: Wuhan Univ, Key Lab Biomed Polymers, Minist Educ, Wuhan 430072, Peoples R China

Wang, Qing-Rong
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h-index: 0
机构:
Wuhan Univ, Key Lab Biomed Polymers, Minist Educ, Wuhan 430072, Peoples R China Wuhan Univ, Key Lab Biomed Polymers, Minist Educ, Wuhan 430072, Peoples R China

Zhuo, Ren-Xi
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机构: Wuhan Univ, Key Lab Biomed Polymers, Minist Educ, Wuhan 430072, Peoples R China

Zhang, Xian-Zheng
论文数: 0 引用数: 0
h-index: 0
机构: Wuhan Univ, Key Lab Biomed Polymers, Minist Educ, Wuhan 430072, Peoples R China
机构:
[1] Wuhan Univ, Key Lab Biomed Polymers, Minist Educ, Wuhan 430072, Peoples R China
基金:
中国国家自然科学基金;
关键词:
MATRIX METALLOPROTEINASES;
CELL DEATH;
THERAPY;
NANOCARRIERS;
DESIGN;
NANOPARTICLES;
STRATEGIES;
RELEASE;
PEPTIDE;
D O I:
10.1039/c4cc07563c
中图分类号:
O6 [化学];
学科分类号:
0703 ;
摘要:
Multifunctional Biotin-PEG-b-PLL(Mal)-peptide-DOX polymeric micelles were prepared to selectively eliminate cancer cells. The micelles were able to enhance cancer cell uptake via the receptor-mediated endocytosis and respond to the stimulus of cancer cell excessive secreted protease MMP-2 to release the anticancer drug and induce apoptosis of cancer cells in a targeted manner.
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页码:465 / 468
页数:4
相关论文
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