Synthesis and biological activity of fluorine-containing amino derivatives based on 4-caranethiol

被引：11

作者：

Sudarikov, D. V. ^{[1
]}

Krymskaya, Yu. V. ^{[1
]}

Il'chenko, N. O. ^{[1
]}

Slepukhin, P. A. ^{[2
,3
]}

Rubtsova, S. A. ^{[1
]}

Kutchin, A. V. ^{[1
]}

机构：

[1] Russian Acad Sci, Inst Chem, Komi Sci Ctr, Ural Branch, 48 Ul Pervomaiskaya, Syktyvkar 167982, Russia

[2] Russian Acad Sci, I Ya Postovsky Inst Organ Synth, Ural Branch, 22-20 Ul S Kovalevskoy Akad Skaya, Ekaterinburg 620990, Russia

[3] Ural Fed Univ, 19 Ul Mira, Ekaterinburg 620002, Russia

来源：

RUSSIAN CHEMICAL BULLETIN | 2018年 / 67卷 / 04期

基金：

俄罗斯基础研究基金会;

关键词：

4-caranethiol; sulfenimines; sulfinimines; chiral fluorine-containing N-substituted alpha-branched sulfinamides; Ruppert-Prakash reagent; fluorine-containing Reformatsky reagent; antimicrobial activity; ASYMMETRIC-SYNTHESIS; STEREOSELECTIVE-SYNTHESIS; TERT-BUTANESULFINIMINES; MEDICINAL CHEMISTRY; CHIRAL AUXILIARY; BETA-PEPTIDES; ACIDS; SULFINIMINES; IMINES; TRIFLUOROPYRUVATE;

D O I：

10.1007/s11172-018-2130-7

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Fluorine-containing N-substituted sulfinamides were synthesized via 4-caranethiol-based sulfenimines and sulfinimines. Stereochemical features of oxidation of sulfenimines and addition of fluorine-containing reagents to sulfinimines were discussed. Antimicrobial activities of the obtained compounds were screened.

引用

页码：731 / 742

页数：12

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