Structure-based design of novel bicyclic nonpeptide inhibitors for the Src SH2 domain

被引:27
|
作者
Shakespeare, WC [1 ]
Bohacek, RS [1 ]
Azimioara, MD [1 ]
Macek, KJ [1 ]
Luke, GP [1 ]
Dalgarno, DC [1 ]
Hatada, MH [1 ]
Lu, XD [1 ]
Violette, SM [1 ]
Bartlett, C [1 ]
Sawyer, TK [1 ]
机构
[1] ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA
关键词
D O I
10.1021/jm0003337
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:3815 / 3819
页数:5
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