Structure-based design of novel bicyclic nonpeptide inhibitors for the Src SH2 domain

被引：28

作者：

Shakespeare, WC ^{[1
]}

Bohacek, RS ^{[1
]}

Azimioara, MD ^{[1
]}

Macek, KJ ^{[1
]}

Luke, GP ^{[1
]}

Dalgarno, DC ^{[1
]}

Hatada, MH ^{[1
]}

Lu, XD ^{[1
]}

Violette, SM ^{[1
]}

Bartlett, C ^{[1
]}

Sawyer, TK ^{[1
]}

机构：

[1] ARIAD Pharmaceut Inc, Cambridge, MA 02139 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2000年 / 43卷 / 21期

关键词：

D O I：

10.1021/jm0003337

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：3815 / 3819

页数：5

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