Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 1. Receptor interactions

被引:357
作者
Jordan, VC [1 ]
机构
[1] Northwestern Univ, Feinberg Sch Med, Roberg H Lurie Comprehens Canc Ctr, Chicago, IL 60611 USA
关键词
D O I
10.1021/jm020449y
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:883 / 908
页数:26
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共 360 条
[61]   Exploring the role of sex steroids through studies of receptor deficient mice [J].
Couse, JF ;
Korach, KS .
JOURNAL OF MOLECULAR MEDICINE-JMM, 1998, 76 (07) :497-511
[62]   4-Hydroxytamoxifen binds to and deactivates the estrogen-related receptor γ [J].
Coward, P ;
Lee, D ;
Hull, MV ;
Lehmann, JM .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2001, 98 (15) :8880-8884
[63]   Estrogen receptors alpha and beta form heterodimers on DNA [J].
Cowley, SM ;
Hoare, S ;
Mosselman, S ;
Parker, MG .
JOURNAL OF BIOLOGICAL CHEMISTRY, 1997, 272 (32) :19858-19862
[64]   The effect of raloxifene on risk of breast cancer in postmenopausal women - Results from the MORE randomized trial [J].
Cummings, SR ;
Eckert, S ;
Krueger, KA ;
Grady, D ;
Powles, TJ ;
Cauley, JA ;
Norton, L ;
Nickelsen, T ;
Bjarnason, NH ;
Morrow, M ;
Lippman, ME ;
Black, D ;
Glusman, JE ;
Costa, A ;
Jordan, VC .
JAMA-JOURNAL OF THE AMERICAN MEDICAL ASSOCIATION, 1999, 281 (23) :2189-2197
[65]   NOVEL ESTROGEN RESPONSE ELEMENTS IDENTIFIED BY GENETIC SELECTION IN YEAST ARE DIFFERENTIALLY RESPONSIVE TO ESTROGENS AND ANTIESTROGENS IN MAMMALIAN-CELLS [J].
DANA, SL ;
HOENER, PA ;
WHEELER, DA ;
LAWRENCE, CB ;
MCDONNELL, DP .
MOLECULAR ENDOCRINOLOGY, 1994, 8 (09) :1193-1207
[66]   IDENTIFICATION OF A CONSERVED REGION REQUIRED FOR HORMONE DEPENDENT TRANSCRIPTIONAL ACTIVATION BY STEROID-HORMONE RECEPTORS [J].
DANIELIAN, PS ;
WHITE, R ;
LEES, JA ;
PARKER, MG .
EMBO JOURNAL, 1992, 11 (03) :1025-1033
[67]  
DAUVOIS S, 1993, J CELL SCI, V106, P1377
[68]   ANTIESTROGEN ICI-164,384 REDUCES CELLULAR ESTROGEN-RECEPTOR CONTENT BY INCREASING ITS TURNOVER [J].
DAUVOIS, S ;
DANIELIAN, PS ;
WHITE, R ;
PARKER, MG .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1992, 89 (09) :4037-4041
[69]   AIB1 is a conduit for kinase-mediated growth factor signaling to the estrogen receptor [J].
de Mora, JF ;
Brown, M .
MOLECULAR AND CELLULAR BIOLOGY, 2000, 20 (14) :5041-5047
[70]   Modifications of benzylphenoxy ethanamine antiestrogen molecules:: Influence affinity for antiestrogen binding site (AEBS) and cell cytotoxicity [J].
Delarue, F ;
Kedjouar, B ;
Mésange, F ;
Bayard, F ;
Faye, JC ;
Poirot, M .
BIOCHEMICAL PHARMACOLOGY, 1999, 57 (06) :657-661