Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 1. Receptor interactions

被引:357
作者
Jordan, VC [1 ]
机构
[1] Northwestern Univ, Feinberg Sch Med, Roberg H Lurie Comprehens Canc Ctr, Chicago, IL 60611 USA
关键词
D O I
10.1021/jm020449y
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:883 / 908
页数:26
相关论文
共 360 条
[1]   OSTEOPOROSIS AFTER OOPHORECTOMY FOR NON-MALIGNANT DISEASE IN PREMENOPAUSAL WOMEN [J].
AITKEN, JM ;
HART, DM ;
ANDERSON, JB ;
LINDSAY, R ;
SMITH, DA ;
SPEIRS, CF .
BRITISH MEDICAL JOURNAL, 1973, 2 (5862) :325-328
[2]   EVIDENCE FOR THE METABOLIC-ACTIVATION OF NON-STEROIDAL ANTIOESTROGENS - A STUDY OF STRUCTURE-ACTIVITY-RELATIONSHIPS [J].
ALLEN, KE ;
CLARK, ER ;
JORDAN, VC .
BRITISH JOURNAL OF PHARMACOLOGY, 1980, 71 (01) :83-91
[3]   Aspartate 351 of estrogen receptor α is not crucial for the antagonist activity of antiestrogens [J].
Anghel, SI ;
Perly, V ;
Melançon, G ;
Barsalou, A ;
Chagnon, S ;
Rosenauer, A ;
Miller, WH ;
Mader, S .
JOURNAL OF BIOLOGICAL CHEMISTRY, 2000, 275 (27) :20867-20872
[4]   Chemoprevention of mammary carcinogenesis in the rat: Combined use of raloxifene and 9-cis-retinoic acid [J].
Anzano, MA ;
Peer, CW ;
Smith, JM ;
Mullen, LT ;
Shrader, MW ;
Logsdon, DL ;
Driver, CL ;
Brown, CC ;
Roberts, AB ;
Sporn, MB .
JOURNAL OF THE NATIONAL CANCER INSTITUTE, 1996, 88 (02) :123-125
[5]   AIB1, a steroid receptor coactivator amplified in breast and ovarian cancer [J].
Anzick, SL ;
Kononen, J ;
Walker, RL ;
Azorsa, DO ;
Tanner, MM ;
Guan, XY ;
Sauter, G ;
Kallioniemi, OP ;
Trent, JM ;
Meltzer, PS .
SCIENCE, 1997, 277 (5328) :965-968
[6]   MOLECULAR BASIS FOR DRUG ACTION [J].
ARIENS, EJ ;
SIMONIS, AM .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1964, 16 (03) :137-&
[7]   STIMULATION OF ESTROGEN RECEPTOR-MEDIATED TRANSCRIPTION AND ALTERATION IN THE PHOSPHORYLATION STATE OF THE RAT UTERINE ESTROGEN-RECEPTOR BY ESTROGEN, CYCLIC ADENOSINE-MONOPHOSPHATE, AND INSULIN-LIKE GROWTH FACTOR-I [J].
ARONICA, SM ;
KATZENELLENBOGEN, BS .
MOLECULAR ENDOCRINOLOGY, 1993, 7 (06) :743-752
[8]   A realistic clinical perspective of tamoxifen and endometrial carcinogenesis [J].
Assikis, VJ ;
Neven, P ;
Jordan, VC ;
Vergote, I .
EUROPEAN JOURNAL OF CANCER, 1996, 32A (09) :1464-1476
[9]  
BARNES LE, 1962, FERTIL STERIL, V13, P472
[10]   Hormone replacement therapy, heart disease, and other considerations [J].
Barrett-Connor, E ;
Grady, D .
ANNUAL REVIEW OF PUBLIC HEALTH, 1998, 19 :55-72