Signaling Bias and Antagonism of Pilocarpine for M3 Muscarinic Acetylcholine Receptor

被引:0
|
作者
Pronin, Alexey N.
Wang, Kelly
Slepak, Vladlen Z.
机构
来源
FASEB JOURNAL | 2018年 / 32卷 / 01期
基金
美国国家卫生研究院;
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
555.7
引用
收藏
页数:2
相关论文
共 50 条
  • [1] Teaching an Old Drug New Tricks: Agonism, Antagonism, and Biased Signaling of Pilocarpine through M3 Muscarinic Acetylcholine Receptor
    Pronin, Alexey N.
    Wang, Qiang
    Slepak, Vladlen Z.
    MOLECULAR PHARMACOLOGY, 2017, 92 (05) : 601 - 612
  • [2] Structure and dynamics of the M3 muscarinic acetylcholine receptor
    Andrew C. Kruse
    Jianxin Hu
    Albert C. Pan
    Daniel H. Arlow
    Daniel M. Rosenbaum
    Erica Rosemond
    Hillary F. Green
    Tong Liu
    Pil Seok Chae
    Ron O. Dror
    David E. Shaw
    William I. Weis
    Jürgen Wess
    Brian K. Kobilka
    Nature, 2012, 482 : 552 - 556
  • [3] m3 muscarinic acetylcholine receptor regulation in the airway
    Billington, CK
    Penn, RB
    AMERICAN JOURNAL OF RESPIRATORY CELL AND MOLECULAR BIOLOGY, 2002, 26 (03) : 269 - 272
  • [4] Structure and dynamics of the M3 muscarinic acetylcholine receptor
    Kruse, Andrew C.
    Hu, Jianxin
    Pan, Albert C.
    Arlow, Daniel H.
    Rosenbaum, Daniel M.
    Rosemond, Erica
    Green, Hillary F.
    Liu, Tong
    Chae, Pil Seok
    Dror, Ron O.
    Shaw, David E.
    Weis, William I.
    Wess, Juergen
    Kobilka, Brian K.
    NATURE, 2012, 482 (7386) : 552 - 556
  • [5] M3 muscarinic acetylcholine receptor in cardiology and oncology
    Patane, Salvatore
    INTERNATIONAL JOURNAL OF CARDIOLOGY, 2014, 177 (02) : 646 - 649
  • [6] Activation State of the M3 Muscarinic Acetylcholine Receptor Modulates Mammalian Odorant Receptor Signaling
    Li, Yun Rose
    Matsunami, Hiroaki
    SCIENCE SIGNALING, 2011, 4 (155)
  • [7] M3 muscarinic acetylcholine receptor-mediated signaling is regulated by distinct mechanisms
    Luo, Jiansong
    Busillo, John M.
    Benovic, Jeffrey L.
    MOLECULAR PHARMACOLOGY, 2008, 74 (02) : 338 - 347
  • [8] The Role of Muscarinic Acetylcholine Receptor M3 in Cardiovascular Diseases
    Liu, Xinxing
    Yu, Yi
    Zhang, Haiying
    Zhang, Min
    Liu, Yan
    INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2024, 25 (14)
  • [9] Roles of M3 muscarinic acetylcholine receptor on gastric functions
    Aihara, T
    Fujishita, T
    Okabe, S
    Matsui, M
    Taketo, M
    JAPANESE JOURNAL OF PHARMACOLOGY, 2002, 88 : 101P - 101P
  • [10] The M3 Muscarinic Acetylcholine Receptor Promotes Epidermal Differentiation
    Duan, Junyan
    Grando, Charles
    Liu, Shuman
    Chernyavsky, Alex
    Chen, Jefferson K.
    Andersen, Bogi
    Grando, Sergei A.
    JOURNAL OF INVESTIGATIVE DERMATOLOGY, 2022, 142 (12) : 3211 - +