3-Nitropyrimido[1,2-a]benzimidazol-4-ones: synthesis and study of alkylation reaction

被引：8

作者：

Fedotov, Victor V. ^{[1
]}

Ulomskiy, Eugeny N. ^{[1
]}

Gorbunov, Evgeny B. ^{[2
]}

Eltsov, Oleg S. ^{[1
]}

Voinkov, Egor K. ^{[1
]}

Savateev, Konstantin V. ^{[1
]}

Drokin, Roman A. ^{[1
]}

Kotovskaya, Svetlana K. ^{[1
]}

Rusinov, Vladimir L. ^{[1
]}

机构：

[1] Ural Fed Univ, 19 Mir St, Ekaterinburg 620002, Russia

[2] Russian Acad Sci, IYa Postovskii Inst Organ Synth, Ural Branch, 22 S Kovalevskoi 20 Akad Skaya St, Ekaterinburg 620990, Russia

来源：

CHEMISTRY OF HETEROCYCLIC COMPOUNDS | 2017年 / 53卷 / 05期

基金：

俄罗斯科学基金会;

关键词：

benzimidazoles; pyrimido[1,2-a]benzimidazol-4-ones; alkylation; stretched-out; SUZUKI-MIYAURA REACTION; PALLADIUM COMPLEXES; DERIVATIVES; MARIBAVIR;

D O I：

10.1007/s10593-017-2095-8

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The reactions of benzimidazol-2-amines with ethyl 3-ethoxy-2-nitroacrylate were used to synthesize a series of pyrimido[1,2-a]-benzimidazoles. An alkylation reaction of the obtained compounds was studied.

引用

页码：582 / 588

页数：7

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