Synthesis of 5-membered ring-type compounds as potential cholecystokinin receptor ligands

被引：0

作者：

Pentassuglia, G ^{[1
]}

Araldi, GL ^{[1
]}

Donati, D ^{[1
]}

Feriani, A ^{[1
]}

Oliosi, B ^{[1
]}

Pasquarello, A ^{[1
]}

Ursini, A ^{[1
]}

机构：

[1] Glaxo SpA, Med Res Ctr, I-37135 Verona, Italy

来源：

FARMACO | 1997年 / 52卷 / 10期

关键词：

D O I：

暂无

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

Imidazolidine-2,4-diones and 1,5-diphenyl tetramic acid derivatives were selected in order to evaluate some 5-membered heterocyclic ring compounds as potential templates for the synthesis of CCK receptor ligands. All the compounds were evaluated in vitro towards both CCK-B and CCK-A receptors.

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页码：573 / 581

页数：9

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