Aluminum dodecatungstophosphate promoted synthesis of 1,5-benzodiazepine derivatives under solvent-free conditions

被引：13

作者：

Fazaeli, Razieh ^{[1
]}

Aliyan, Hamid

Tangestaninejad, Shahram

机构：

[1] Islamic Azad Univ, Dept Chem, Shahreza Branch, Shahreza 86145311, Iran

[2] Isfahan Univ, Dept Chem, Esfahan 8174673441, Iran

来源：

HETEROCYCLES | 2007年 / 71卷 / 04期

关键词：

D O I：

10.3987/COM-06-10948

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Solid heteropoly acids (A1TP and A1MP) are easily used as efficient catalyst for conversion of o-phenylenediamines and ketones to their corresponding 2,3-dihydro-1H-1,5-benzodiazepines at room temperature under solvent-free conditions. The method is an easy, rapid, and high yielding reaction for the synthesis of 1,5-benzodiazepine derivatives and is applicable to both cyclic or acyclic ketones without significant difference.

引用

页码：805 / 814

页数：10

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