Synthesis of Terpenoid-Like Bischalcones from α- and β-Ionones and Their Biological Activities

被引：5

作者：

Findik, Esra ^{[1
]}

Dingil, Alparslan ^{[1
]}

Karaman, Isa ^{[2
]}

Ceylan, Mustafa ^{[1
]}

机构：

[1] Gaziosmanpasa Univ, Dept Chem, Fac Arts & Sci, TR-60250 Tokat, Turkey

[2] Gaziosmanpasa Univ, Dept Biol, Fac Arts & Sci, TR-60250 Tokat, Turkey

来源：

SYNTHETIC COMMUNICATIONS | 2009年 / 39卷 / 24期

关键词：

Antibacterial and antifungal activity; terpenoid-like bischalcone; BIOEVALUATION; LEISHMANIASIS; CHEMOTHERAPY; PYRIMIDINES;

D O I：

10.1080/00397910902900696

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Ionone-based terpenoid-like bischalcones (3a-h and 4a-h) were synthesized from the reaction of alpha- and/or beta-ionones with aldehyde derivatives in excellent yields. The antibacterial activities of synthesized compounds were screened against human pathogenic micro-organisms by employing the disk-diffusion technique.

引用

页码：4362 / 4374

页数：13

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