Synthesis of benzonaphtho[1,4]diazepine derivatives via the reaction of 2-aminoarylbenzimidamides with 2,3-dichloro-1,4-naphthoquinone

被引：13

作者：

El-Shaieb, Kamal M. ^{[1
]}

机构：

[1] Menia Univ, Dept Chem, Fac Sci, El Minia, Egypt

来源：

JOURNAL OF CHEMICAL RESEARCH | 2010年 / 03期

关键词：

aminobenzimidamides; naphthoquinone; CT-complexes; benzonaphthodiazepines; BIOLOGICAL EVALUATION; ANTIPLATELET; INHIBITORS; AFFINITY;

D O I：

10.3184/030823410X12659615450519

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A series of (Z)-13-(arylimino)-12,13-dihydro-5H-benzo[e]naphtho[2,3-b][1,4]diazepine-6,11-dione derivatives have been synthesised by one pot cyclisation in good yield via electron donor-acceptor complexes by reacting 2-amino-arylbenzimidamides with 2,3-dichloro-1,4-naphthoquinone. The high yield and simplified workup procedure in addition to the mild and neutral reaction conditions are the main advantages of this approach.

引用

页码：137 / 139

页数：3

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