Recent Advances in the Discovery of Competitive Protein Tyrosine Phosphatase 1B Inhibitors for the Treatment of Diabetes, Obesity, and Cancer

被引：305

作者：

Combs, Andrew P. ^{[1
]}

机构：

[1] Incyte Corp, Expt Stn, Wilmington, DE 19880 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2010年 / 53卷 / 06期

关键词：

STRUCTURE-BASED DESIGN; INSULIN SENSITIVITY; STRUCTURAL BASIS; TC-PTP; POTENT; ACIDS; IDENTIFICATION; SITE;

D O I：

10.1021/jm901090b

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：2333 / 2344

页数：12

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