COMBINATION OF SORAFENIB AND 5-AZACYTIDINE HAS SIGNIFICANT ACTIVITY IN PATIENTS WITH RELAPSED/REFRACTORY OR UNTREATED ACUTE MYELOID LEUKEMIA AND FLT3-ITD MUTATION

被引:0
|
作者
Ravandi, Farhad [1 ]
Alattar, Mona Lisa [1 ]
Levis, Mark [1 ]
Garcia-Manero, Guillermo [1 ]
Richie, Mary A. [1 ]
Daver, Naval [1 ]
Faderl, Stefan [1 ]
Borthakur, Gautam [1 ]
Burger, Jan [1 ]
Kadia, Tapan [1 ]
Grunwald, Michael [1 ]
Dellasala, Sara [1 ]
Cortes, Jorge [1 ]
Kantarjian, Hagop [1 ]
机构
[1] Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA
关键词
D O I
暂无
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
45
引用
收藏
页码:S19 / S20
页数:2
相关论文
共 50 条
  • [41] Pyruvate Dehydrogenase (PDH) Activity Is a Source of Resistance to Sorafenib in FLT3-ITD Expressing Acute Myeloid Leukemia (AML)
    Anderson, Rebecca G.
    Pladna, Kristin M.
    Pardee, Timothy S.
    BLOOD, 2017, 130
  • [42] Arsenic Trioxide and Sorafenib Induce Synthetic Lethality of FLT3-ITD Acute Myeloid Leukemia Cells
    Wang, Rui
    Li, Ying
    Gong, Ping
    Gabrilove, Janice
    Waxman, Samuel
    Jing, Yongkui
    MOLECULAR CANCER THERAPEUTICS, 2018, 17 (09) : 1871 - 1880
  • [43] NFATC1 MEDIATES SORAFENIB RESISTANCE IN FLT3-ITD POSITIVE ACUTE MYELOID LEUKEMIA
    Michel, C.
    Metzelder, S.
    Bonin, M.
    Rehberger, M.
    Hessmann, E.
    Brendel, C.
    Stiewe, T.
    Ellenrieder, V.
    Haferlach, T.
    Bornhaeuser, M.
    Neubauer, A.
    Burchert, A.
    HAEMATOLOGICA, 2014, 99 : 290 - 290
  • [44] Decitabine and sorafenib therapy in FLT3-ITD mutant acute myeloid leukemia- A case series
    Muppidi, Monica R.
    Griffiths, Elizabeth A.
    Thompson, James E.
    Ford, Laurie A.
    Freyer, Craig W.
    Wetzler, Meir
    Wang, Eunice S.
    CLINICAL LYMPHOMA MYELOMA & LEUKEMIA, 2015, 15 : S187 - S187
  • [45] FLT3 AND FLT3-ITD GENE MUTATIONS AND PROGNOSIS IN PATIENTS WITH ACUTE MYELOID LEUKEMIA
    Chen, L. G.
    Pei, R. Z.
    Lu, Y.
    Zhang, P. S.
    Liu, X. H.
    Du, X. H.
    Chen, D.
    Cao, J. J.
    Li, S. Y.
    JOURNAL OF BIOLOGICAL REGULATORS AND HOMEOSTATIC AGENTS, 2019, 33 (06) : 1855 - 1861
  • [46] Sorafenib priming may augment salvage chemotherapy in relapsed and refractory FLT3-ITD-positive acute myeloid leukemia
    K D Cummins
    S M Jane
    S Ninkovic
    A Bazargan
    R Filshie
    G Sutrave
    M Hertzberg
    A Scott
    S Lane
    C K Yannakou
    D Ritchie
    J D'Rozario
    J Black
    K Bavishi
    A Wei
    Blood Cancer Journal, 2014, 4 : e237 - e237
  • [47] Sorafenib priming may augment salvage chemotherapy in relapsed and refractory FLT3-ITD-positive acute myeloid leukemia
    Cummins, K. D.
    Jane, S. M.
    Ninkovic, S.
    Bazargan, A.
    Filshie, R.
    Sutrave, G.
    Hertzberg, M.
    Scott, A.
    Lane, S.
    Yannakou, C. K.
    Ritchie, D.
    D'Rozario, J.
    Black, J.
    Bavishi, K.
    Wei, A.
    BLOOD CANCER JOURNAL, 2014, 4 : e237 - e237
  • [48] A novel combination regimen of BET and FLT3 inhibition for FLT3-ITD acute myeloid leukemia
    Lee, Lauren
    Hizukuri, Yoshiyuki
    Severson, Paul
    Powell, Benjamin
    Zhang, Chao
    Ma, Yan
    Narahara, Maiko
    Sumi, Hiroyuki
    Hernandez, Daniela
    Rajkhowa, Trivikram
    Bollag, Gideon
    Levis, Mark
    HAEMATOLOGICA, 2021, 106 (04) : 1022 - 1033
  • [49] A Novel Combination Regimen of BET and FLT3 Inhibition for FLT3-ITD Acute Myeloid Leukemia
    Lee, Lauren
    Hizukuri, Yoshiyuki
    Severson, Paul
    Powell, Ben
    Zhang, Chao
    Ma, Yan
    Narahara, Maiko
    Sumi, Hiroyuki
    Bollag, Gideon
    Levis, Mark J.
    BLOOD, 2019, 134
  • [50] 8-chloro-adenosine activity in FLT3-ITD acute myeloid leukemia
    Buettner, Ralf
    Le Xuan Truong Nguyen
    Kumar, Bijender
    Morales, Corey
    Liu, Chao
    Chen, Lisa S.
    Pemovska, Tea
    Synold, Timothy W.
    Palmer, Joycelynne
    Thompson, Ryan
    Li, Ling
    Dinh Hoa Hoang
    Zhang, Bin
    Ghoda, Lucy
    Kowolik, Claudia
    Kontro, Mika
    Leitch, Calum
    Wennerberg, Krister
    Yu, Xiaochun
    Chen, Ching-Cheng
    Horne, David
    Gandhi, Varsha
    Pullarkat, Vinod
    Marcucci, Guido
    Rosen, Steven T.
    JOURNAL OF CELLULAR PHYSIOLOGY, 2019, 234 (09) : 16295 - 16303