共 23 条
Targeting the mevalonate pathway in multiple myeloma
被引:3
作者:

van der Spek, Ellen
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Med Ctr Utrecht, Dept Hematol, NL-3584 CX Utrecht, Netherlands Univ Med Ctr Utrecht, Dept Hematol, NL-3584 CX Utrecht, Netherlands
机构:
[1] Univ Med Ctr Utrecht, Dept Hematol, NL-3584 CX Utrecht, Netherlands
关键词:
Multiple myeloma;
Mevalonate pathway;
Plasma cell lines;
FPP;
GGPP;
CELL-LINES;
DRUG-RESISTANCE;
PLASMA-CELLS;
APOPTOSIS;
SIMVASTATIN;
INHIBITOR;
SURVIVAL;
PROTEIN;
GERANYLGERANYLATION;
FARNESYLATION;
D O I:
10.1016/j.leukres.2009.07.027
中图分类号:
R73 [肿瘤学];
学科分类号:
100214 ;
摘要:
引用
收藏
页码:267 / 268
页数:2
相关论文
共 23 条
[1]
Farnesyltransferase inhibitor tipifarnib is well tolerated, induces stabilization of disease, and inhibits farnesylation and oncogenic/tumor survival pathways in patients with advanced multiple myeloma
[J].
Alsina, M
;
Fonseca, R
;
Wilson, EF
;
Belle, AN
;
Gerbino, E
;
Price-Troska, T
;
Overton, RM
;
Ahmann, G
;
Bruzek, LM
;
Adjei, AA
;
Kaufmann, SH
;
Wright, JJ
;
Sullivan, D
;
Djulbegovic, B
;
Cantor, AB
;
Greipp, PR
;
Dalton, WS
;
Sebti, SM
.
BLOOD,
2004, 103 (09)
:3271-3277

Alsina, M
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Fonseca, R
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Wilson, EF
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Belle, AN
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Gerbino, E
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Price-Troska, T
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Overton, RM
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Ahmann, G
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Bruzek, LM
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Adjei, AA
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Kaufmann, SH
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Wright, JJ
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Sullivan, D
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Djulbegovic, B
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Cantor, AB
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Greipp, PR
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Dalton, WS
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA

Sebti, SM
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, MRCDRDIS,Drug Discovery Program, Tampa, FL 33612 USA
[2]
Maintenance, therapy with thalidomide improves survival in patients with multiple myeloma
[J].
Attal, Michel
;
Harousseau, Jean-Luc
;
Leyvraz, Serge
;
Doyen, Chantal
;
Hulin, Cyrille
;
Benboubker, Lofti
;
Agha, Ibrahim Yakoub
;
Bourhis, Jean-Henri
;
Garderet, Laurent
;
Pegourie, Brigitte
;
Dumontet, Charles
;
Renaud, Marc
;
Voillat, Laurent
;
Berthou, Christian
;
Marit, Gerald
;
Monconduit, Mathieu
;
Caillot, Denis
;
Grobois, Bernard
;
Avet-Loiseau, Herve
;
Moreau, Philippe
;
Facon, Thierry
.
BLOOD,
2006, 108 (10)
:3289-3294

Attal, Michel
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Harousseau, Jean-Luc
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Leyvraz, Serge
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Doyen, Chantal
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Hulin, Cyrille
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Benboubker, Lofti
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Agha, Ibrahim Yakoub
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Bourhis, Jean-Henri
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Garderet, Laurent
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Pegourie, Brigitte
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Dumontet, Charles
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Renaud, Marc
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Voillat, Laurent
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Berthou, Christian
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Marit, Gerald
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Monconduit, Mathieu
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Caillot, Denis
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Grobois, Bernard
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Avet-Loiseau, Herve
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Moreau, Philippe
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France

Facon, Thierry
论文数: 0 引用数: 0
h-index: 0
机构: Hop Purpan, Dept Hematol, Toulouse, France
[3]
Efficacy of pamidronate in reducing skeletal events in patients with advanced multiple myeloma
[J].
Berenson, JR
;
Lichtenstein, A
;
Porter, L
;
Dimopoulos, MA
;
Bordoni, R
;
George, S
;
Lipton, A
;
Keller, A
;
Ballester, O
;
Kovacs, MJ
;
Blacklock, HA
;
Bell, R
;
Simeone, J
;
Reitsma, DJ
;
Heffernan, M
;
Seaman, J
;
Knight, RD
.
NEW ENGLAND JOURNAL OF MEDICINE,
1996, 334 (08)
:488-493

Berenson, JR
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Lichtenstein, A
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Porter, L
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Dimopoulos, MA
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Bordoni, R
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

George, S
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Lipton, A
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Keller, A
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Ballester, O
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Kovacs, MJ
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Blacklock, HA
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Bell, R
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Simeone, J
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Reitsma, DJ
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Heffernan, M
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Seaman, J
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024

Knight, RD
论文数: 0 引用数: 0
h-index: 0
机构: UNIV CALIF LOS ANGELES,JONSSON COMPREHENS CANC CTR,SCH MED,LOS ANGELES,CA 90024
[4]
The farnesyl transferase inhibitor, FTI-277, inhibits growth and induces apoptosis in drug-resistant myeloma tumor cells
[J].
Bolick, SCE
;
Landowski, TH
;
Boulware, D
;
Oshiro, MM
;
Ohkanda, J
;
Hamilton, AD
;
Sebti, SD
;
Dalton, WS
.
LEUKEMIA,
2003, 17 (02)
:451-457

Bolick, SCE
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL 33612 USA

Landowski, TH
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL 33612 USA

Boulware, D
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL 33612 USA

Oshiro, MM
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL 33612 USA

Ohkanda, J
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL 33612 USA

Hamilton, AD
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL 33612 USA

Sebti, SD
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL 33612 USA

Dalton, WS
论文数: 0 引用数: 0
h-index: 0
机构: Univ S Florida, Coll Med, H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL 33612 USA
[5]
Statins activate the mitochondrial pathway of apoptosis in human lymphoblasts and myeloma cells
[J].
Cafforio, P
;
Dammacco, F
;
Gernone, A
;
Silvestris, F
.
CARCINOGENESIS,
2005, 26 (05)
:883-891

论文数: 引用数:
h-index:
机构:

Dammacco, F
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Bari, Dept Internal Med & Oncol, I-70124 Bari, Italy Univ Bari, Dept Internal Med & Oncol, I-70124 Bari, Italy

Gernone, A
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Bari, Dept Internal Med & Oncol, I-70124 Bari, Italy Univ Bari, Dept Internal Med & Oncol, I-70124 Bari, Italy

论文数: 引用数:
h-index:
机构:
[6]
Statins synergistically potentiate 7-hydroxystaurosporine (UCN-01) lethality in human leukemia and myeloma cells by disrupting Ras farnesylation and activation
[J].
Dai, Yun
;
Khanna, Payal
;
Chen, Shuang
;
Pei, Xin-Yan
;
Dent, Paul
;
Grant, Steven
.
BLOOD,
2007, 109 (10)
:4415-4423

Dai, Yun
论文数: 0 引用数: 0
h-index: 0
机构: Virginia Commonwealth Univ, Med Coll Virginia, Massey Canc Ctr, Dept Med,Div Hematol Oncol, Richmond, VA 23298 USA

Khanna, Payal
论文数: 0 引用数: 0
h-index: 0
机构: Virginia Commonwealth Univ, Med Coll Virginia, Massey Canc Ctr, Dept Med,Div Hematol Oncol, Richmond, VA 23298 USA

Chen, Shuang
论文数: 0 引用数: 0
h-index: 0
机构: Virginia Commonwealth Univ, Med Coll Virginia, Massey Canc Ctr, Dept Med,Div Hematol Oncol, Richmond, VA 23298 USA

Pei, Xin-Yan
论文数: 0 引用数: 0
h-index: 0
机构: Virginia Commonwealth Univ, Med Coll Virginia, Massey Canc Ctr, Dept Med,Div Hematol Oncol, Richmond, VA 23298 USA

Dent, Paul
论文数: 0 引用数: 0
h-index: 0
机构: Virginia Commonwealth Univ, Med Coll Virginia, Massey Canc Ctr, Dept Med,Div Hematol Oncol, Richmond, VA 23298 USA

Grant, Steven
论文数: 0 引用数: 0
h-index: 0
机构: Virginia Commonwealth Univ, Med Coll Virginia, Massey Canc Ctr, Dept Med,Div Hematol Oncol, Richmond, VA 23298 USA
[7]
REGULATION OF THE MEVALONATE PATHWAY
[J].
GOLDSTEIN, JL
;
BROWN, MS
.
NATURE,
1990, 343 (6257)
:425-430

GOLDSTEIN, JL
论文数: 0 引用数: 0
h-index: 0
机构:
UNIV TEXAS, SW MED CTR, DEPT INTERNAL MED, DALLAS, TX 75235 USA UNIV TEXAS, SW MED CTR, DEPT INTERNAL MED, DALLAS, TX 75235 USA

BROWN, MS
论文数: 0 引用数: 0
h-index: 0
机构:
UNIV TEXAS, SW MED CTR, DEPT INTERNAL MED, DALLAS, TX 75235 USA UNIV TEXAS, SW MED CTR, DEPT INTERNAL MED, DALLAS, TX 75235 USA
[8]
The effect of statin use at the time of autologous transplant on response and survival in multiple myeloma
[J].
Hamadani, Mehdi
;
Hade, Erinn
;
Benson, Don M.
;
Hofineister, Craig C.
.
BIOLOGY OF BLOOD AND MARROW TRANSPLANTATION,
2008, 14 (03)
:351-352

论文数: 引用数:
h-index:
机构:

Hade, Erinn
论文数: 0 引用数: 0
h-index: 0
机构:
Ohio State Univ, Arthur G James Canc Hosp, Div Hematol & Oncol, Columbus, OH 43210 USA Ohio State Univ, Arthur G James Canc Hosp, Div Hematol & Oncol, Columbus, OH 43210 USA

Benson, Don M.
论文数: 0 引用数: 0
h-index: 0
机构:
Ohio State Univ, Arthur G James Canc Hosp, Div Hematol & Oncol, Columbus, OH 43210 USA Ohio State Univ, Arthur G James Canc Hosp, Div Hematol & Oncol, Columbus, OH 43210 USA

Hofineister, Craig C.
论文数: 0 引用数: 0
h-index: 0
机构:
Ohio State Univ, Arthur G James Canc Hosp, Div Hematol & Oncol, Columbus, OH 43210 USA Ohio State Univ, Arthur G James Canc Hosp, Div Hematol & Oncol, Columbus, OH 43210 USA
[9]
Sterol-independent regulation of 3-hydroxy-3-methylglutaryl coenzyme A reductase in tumor cells
[J].
Hentosh, P
;
Yuh, SH
;
Elson, CE
;
Peffley, DM
.
MOLECULAR CARCINOGENESIS,
2001, 32 (03)
:154-166

Hentosh, P
论文数: 0 引用数: 0
h-index: 0
机构: Univ Hlth Sci, Dept Pharmacol, Kansas City, MO USA

Yuh, SH
论文数: 0 引用数: 0
h-index: 0
机构: Univ Hlth Sci, Dept Pharmacol, Kansas City, MO USA

Elson, CE
论文数: 0 引用数: 0
h-index: 0
机构: Univ Hlth Sci, Dept Pharmacol, Kansas City, MO USA

Peffley, DM
论文数: 0 引用数: 0
h-index: 0
机构: Univ Hlth Sci, Dept Pharmacol, Kansas City, MO USA
[10]
Risk of multiple myeloma following medication use and medical conditions: A case-control study in Connecticut women
[J].
Landgren, Ola
;
Zhang, Yawei
;
Zahm, Sheila Hoar
;
Inskip, Peter
;
Zheng, Tongzhang
;
Baris, Dalsu
.
CANCER EPIDEMIOLOGY BIOMARKERS & PREVENTION,
2006, 15 (12)
:2342-2347

Landgren, Ola
论文数: 0 引用数: 0
h-index: 0
机构: NCI, Div Canc Epidemiol & Genet, Genet Epidemiol Branch, NIH,Dept Hlth & Human Serv, Bethesda, MD 20892 USA

Zhang, Yawei
论文数: 0 引用数: 0
h-index: 0
机构: NCI, Div Canc Epidemiol & Genet, Genet Epidemiol Branch, NIH,Dept Hlth & Human Serv, Bethesda, MD 20892 USA

Zahm, Sheila Hoar
论文数: 0 引用数: 0
h-index: 0
机构: NCI, Div Canc Epidemiol & Genet, Genet Epidemiol Branch, NIH,Dept Hlth & Human Serv, Bethesda, MD 20892 USA

Inskip, Peter
论文数: 0 引用数: 0
h-index: 0
机构: NCI, Div Canc Epidemiol & Genet, Genet Epidemiol Branch, NIH,Dept Hlth & Human Serv, Bethesda, MD 20892 USA

Zheng, Tongzhang
论文数: 0 引用数: 0
h-index: 0
机构: NCI, Div Canc Epidemiol & Genet, Genet Epidemiol Branch, NIH,Dept Hlth & Human Serv, Bethesda, MD 20892 USA

Baris, Dalsu
论文数: 0 引用数: 0
h-index: 0
机构: NCI, Div Canc Epidemiol & Genet, Genet Epidemiol Branch, NIH,Dept Hlth & Human Serv, Bethesda, MD 20892 USA