Copper-mediated cross-coupling reactions of N-unsubstituted sulfoximines and aryl halides

被引:101
作者
Cho, GY [1 ]
Rémy, P [1 ]
Jansson, J [1 ]
Moessner, C [1 ]
Bolm, C [1 ]
机构
[1] Univ Aachen, Rhein Westfal TH Aachen, Inst Organ Chem, D-52056 Aachen, Germany
关键词
D O I
10.1021/ol048806h
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Copper-mediated cross-coupling reactions of sulfoximines with aryl iodides and aryl bromides provide N-arylated sulfoximines in high yields. The method is complementary to the known palladium-catalyzed N-arylation and allows the preparation of N-arylated sulfoximines, which have previously been inaccessible.
引用
收藏
页码:3293 / 3296
页数:4
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