Pyrrolo [3,4-e][1,2,3]triazolo[1,5-a]pyrimidine and pyrrolo[3,4-d][1,2,3]triazolo[1,5-a]pyrimidine.: New tricyclic ring systems of biological interest

被引：27

作者：

Lauria, A ^{[1
]}

Diana, P ^{[1
]}

Barraja, P ^{[1
]}

Almerico, AM ^{[1
]}

Cirrincione, G ^{[1
]}

Dattolo, G ^{[1
]}

机构：

[1] Univ Palermo, Dipartimento Farmacochim Tossicol & Biol, I-90123 Palermo, Italy

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2000年 / 37卷 / 04期

关键词：

D O I：

10.1002/jhet.5570370413

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Derivatives of the new ring system pyrrolo[3,4-e][1,2,3] triazolo[1,5-a]pyrimidine 6 were prepared in high yields in one step by reaction of 3-azidopyrrole 3 and substituted acetonitriles. Compound 6b rearranged, upon heating in dimethyl sulfoxide in the presence of water, to pyrrolo[3,4-d]1,2,3]triazolo[1,5-a]pyrimidine 7.

引用

页码：747 / 750

页数：4

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