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- [21] Autophagy dictates sensitivity to PRMT5 inhibitor in breast cancerScientific Reports, 13Charles Brobbey论文数: 0 引用数: 0 h-index: 0机构: Medical University of South Carolina,Department of Biochemistry and Molecular BiologyShasha Yin论文数: 0 引用数: 0 h-index: 0机构: Medical University of South Carolina,Department of Biochemistry and Molecular BiologyLiu Liu论文数: 0 引用数: 0 h-index: 0机构: Medical University of South Carolina,Department of Biochemistry and Molecular BiologyLauren E. Ball论文数: 0 引用数: 0 h-index: 0机构: Medical University of South Carolina,Department of Biochemistry and Molecular BiologyPhilip H. Howe论文数: 0 引用数: 0 h-index: 0机构: Medical University of South Carolina,Department of Biochemistry and Molecular BiologyJoe R. Delaney论文数: 0 引用数: 0 h-index: 0机构: Medical University of South Carolina,Department of Biochemistry and Molecular BiologyWenjian Gan论文数: 0 引用数: 0 h-index: 0机构: Medical University of South Carolina,Department of Biochemistry and Molecular Biology
- [22] Identification of a CARM1 Inhibitor with Potent In Vitro and In Vivo Activity in Preclinical Models of Multiple MyelomaScientific Reports, 7Allison E. Drew论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitOscar Moradei论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitSuzanne L. Jacques论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitNathalie Rioux论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitAnn P. Boriack-Sjodin论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitChristina Allain论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitMargaret Porter Scott论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitLei Jin论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitAlejandra Raimondi论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitJessica L. Handler论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitHeidi M. Ott论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitRyan G. Kruger论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitMichael T. McCabe论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitChristopher Sneeringer论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitThomas Riera论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitGideon Shapiro论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitNigel J. Waters论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitLorna H. Mitchell论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitKenneth W. Duncan论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitMikel P. Moyer论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitRobert A. Copeland论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitJesse Smith论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitRichard Chesworth论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance UnitScott A. Ribich论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Epigenetics Discovery Performance Unit
- [23] Identification of a CARM1 Inhibitor with Potent In Vitro and In Vivo Activity in Preclinical Models of Multiple MyelomaSCIENTIFIC REPORTS, 2017, 7Drew, Allison E.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USAMoradei, Oscar论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USAJacques, Suzanne L.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USARioux, Nathalie论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USABoriack-Sjodin, Ann P.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USAAllain, Christina论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USAScott, Margaret Porter论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USAJin, Lei论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USARaimondi, Alejandra论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USAHandler, Jessica L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Epigenet Discovery Performance Unit, Oncol R&D, Collegeville, PA USA Epizyme Inc, Cambridge, MA 02139 USAOtt, Heidi M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Epigenet Discovery Performance Unit, Oncol R&D, Collegeville, PA USA Epizyme Inc, Cambridge, MA 02139 USAKruger, Ryan G.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Epigenet Discovery Performance Unit, Oncol R&D, Collegeville, PA USA Epizyme Inc, Cambridge, MA 02139 USAMcCabe, Michael T.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Epigenet Discovery Performance Unit, Oncol R&D, Collegeville, PA USA Epizyme Inc, Cambridge, MA 02139 USASneeringer, Christopher论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USARiera, Thomas论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USAShapiro, Gideon论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USAWaters, Nigel J.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USAMitchell, Lorna H.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USADuncan, Kenneth W.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USAMoyer, Mikel P.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USACopeland, Robert A.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USASmith, Jesse论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USAChesworth, Richard论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USARibich, Scott A.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USA
- [24] Preclinical characterization of ATG-042-198, a novel MTAP null-selective PRMT5 inhibitorCANCER RESEARCH, 2024, 84 (06)Kong, Ya论文数: 0 引用数: 0 h-index: 0Zhang, Ming论文数: 0 引用数: 0 h-index: 0Jiang, Lulu论文数: 0 引用数: 0 h-index: 0Xu, Ruiting论文数: 0 引用数: 0 h-index: 0Jiang, Bin论文数: 0 引用数: 0 h-index: 0Dai, Guoqiang论文数: 0 引用数: 0 h-index: 0He, Yulong论文数: 0 引用数: 0 h-index: 0Liu, Huiling论文数: 0 引用数: 0 h-index: 0Mei, Jay论文数: 0 引用数: 0 h-index: 0Hou, Bing论文数: 0 引用数: 0 h-index: 0Shan, Bo论文数: 0 引用数: 0 h-index: 0
- [25] PRMT5 Promotes EMT Through Regulating Akt Activity in Human Lung CancerCELL TRANSPLANTATION, 2021, 30Huang, Jianhao论文数: 0 引用数: 0 h-index: 0机构: Nanjing Med Univ, Shanghai East Clin Med Coll, Dept Pulm & Crit Care Med, Nanjing 200120, Peoples R China Tongji Univ, Shanghai East Hosp, Dept Pulm & Crit Care Med, Sch Med, Shanghai 200120, Peoples R China Nanjing Med Univ, Shanghai East Clin Med Coll, Dept Pulm & Crit Care Med, Nanjing 200120, Peoples R ChinaZheng, Yonghua论文数: 0 引用数: 0 h-index: 0机构: Tongji Univ Sch Med, Shanghai East Hosp, Dept Pulm & Crit Care Med, Shanghai, Peoples R China Nanjing Med Univ, Shanghai East Clin Med Coll, Dept Pulm & Crit Care Med, Nanjing 200120, Peoples R ChinaZheng, Xiao论文数: 0 引用数: 0 h-index: 0机构: Tongji Univ Sch Med, Shanghai East Hosp, Dept Pulm & Crit Care Med, Shanghai, Peoples R China Nanjing Med Univ, Shanghai East Clin Med Coll, Dept Pulm & Crit Care Med, Nanjing 200120, Peoples R ChinaQian, Bao论文数: 0 引用数: 0 h-index: 0机构: Tongji Univ Sch Med, Shanghai East Hosp, Dept Pulm & Crit Care Med, Shanghai, Peoples R China Nanjing Med Univ, Shanghai East Clin Med Coll, Dept Pulm & Crit Care Med, Nanjing 200120, Peoples R ChinaYin, Qi论文数: 0 引用数: 0 h-index: 0机构: Tongji Univ, Shanghai East Hosp, Dept Pulm & Crit Care Med, Sch Med, Shanghai 200120, Peoples R China Nanjing Med Univ, Shanghai East Clin Med Coll, Dept Pulm & Crit Care Med, Nanjing 200120, Peoples R ChinaLu, Jingjing论文数: 0 引用数: 0 h-index: 0机构: Tongji Univ, Shanghai East Hosp, Dept Pulm & Crit Care Med, Sch Med, Shanghai 200120, Peoples R China Nanjing Med Univ, Shanghai East Clin Med Coll, Dept Pulm & Crit Care Med, Nanjing 200120, Peoples R ChinaLei, Han论文数: 0 引用数: 0 h-index: 0机构: Nanjing Med Univ, Shanghai East Clin Med Coll, Dept Pulm & Crit Care Med, Nanjing 200120, Peoples R China Nanjing Med Univ, Shanghai East Clin Med Coll, Dept Pulm & Crit Care Med, Nanjing 200120, Peoples R China
- [26] The discovery and preclinical characterization of the MTA cooperative PRMT5 inhibitor AM-9747CANCER RESEARCH, 2022, 82 (12)Belmontes, Brian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USAPolicheni, Antonia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USALiu, Siyuan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USASlemmons, Katherine论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USAMoriguchi, Jodi论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USAMa, Hayley论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USAAiello, Daniel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USAYang, Yajing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USAVestergaard, Mikkel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Copenhagen, Denmark Amgen Inc, Thousand Oaks, CA USACowland, Sanne论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Copenhagen, Denmark Amgen Inc, Thousand Oaks, CA USAAnderson, Jan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Copenhagen, Denmark Amgen Inc, Thousand Oaks, CA USASarvary, Ian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Copenhagen, Denmark Amgen Inc, Thousand Oaks, CA USATamayo, Nuria论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USAPettus, Liping论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USAMukund, Susmith论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, Thousand Oaks, CA USAPope, Leszek论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USAAllen, Jennifer R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USAGlad, Sanne论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Copenhagen, Denmark Amgen Inc, Thousand Oaks, CA USABourbeau, Matthew论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USAHughes, Paul E.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA USA Amgen Inc, Thousand Oaks, CA USA
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- [29] Structure-Based Discovery and Biological Assays of a Novel PRMT5 Inhibitor for Non-Small Cell Lung CancerMOLECULES, 2022, 27 (21):Chen, Yingqing论文数: 0 引用数: 0 h-index: 0机构: Dalian Univ, Med Coll, Chron Dis Res Ctr, Dalian 116622, Peoples R China Dalian Univ, Med Coll, Chron Dis Res Ctr, Dalian 116622, Peoples R ChinaZhang, Mingyu论文数: 0 引用数: 0 h-index: 0机构: Dalian Univ, Med Coll, Chron Dis Res Ctr, Dalian 116622, Peoples R China Dalian Univ, Med Coll, Chron Dis Res Ctr, Dalian 116622, Peoples R ChinaWu, Anxin论文数: 0 引用数: 0 h-index: 0机构: Dalian Univ, Med Coll, Chron Dis Res Ctr, Dalian 116622, Peoples R China Dalian Univ, Med Coll, Chron Dis Res Ctr, Dalian 116622, Peoples R ChinaYao, Xiaojun论文数: 0 引用数: 0 h-index: 0机构: Macau Univ Sci & Technol, Dr Nehers Biophys Lab Innovat Drug Discovery, State Key Lab Qual Res Chinese Med, Taipa 999078, Macao, Peoples R China Dalian Univ, Med Coll, Chron Dis Res Ctr, Dalian 116622, Peoples R ChinaWang, Qianqian论文数: 0 引用数: 0 h-index: 0机构: Dalian Univ, Med Coll, Chron Dis Res Ctr, Dalian 116622, Peoples R China Dalian Univ, Med Coll, Chron Dis Res Ctr, Dalian 116622, Peoples R China
- [30] Targeting PRMT5 enhances the radiosensitivity of tumor cells grown in vitro and in vivoSCIENTIFIC REPORTS, 2024, 14 (01):Degorre, Charlotte论文数: 0 引用数: 0 h-index: 0机构: NCI, Radiat Oncol Branch, 10 Ctr Dr MSC 1002,Bldg 10,B3B69B, Bethesda, MD 20892 USA NCI, Radiat Oncol Branch, 10 Ctr Dr MSC 1002,Bldg 10,B3B69B, Bethesda, MD 20892 USALohard, Steven论文数: 0 引用数: 0 h-index: 0机构: NCI, Radiat Oncol Branch, 10 Ctr Dr MSC 1002,Bldg 10,B3B69B, Bethesda, MD 20892 USA NCI, Radiat Oncol Branch, 10 Ctr Dr MSC 1002,Bldg 10,B3B69B, Bethesda, MD 20892 USABobrek, Christina N.论文数: 0 引用数: 0 h-index: 0机构: NCI, Radiat Oncol Branch, 10 Ctr Dr MSC 1002,Bldg 10,B3B69B, Bethesda, MD 20892 USA NCI, Radiat Oncol Branch, 10 Ctr Dr MSC 1002,Bldg 10,B3B69B, Bethesda, MD 20892 USARawal, Komal N.论文数: 0 引用数: 0 h-index: 0机构: NCI, Radiat Oncol Branch, 10 Ctr Dr MSC 1002,Bldg 10,B3B69B, Bethesda, MD 20892 USA NCI, Radiat Oncol Branch, 10 Ctr Dr MSC 1002,Bldg 10,B3B69B, Bethesda, MD 20892 USAKuhn, Skyler论文数: 0 引用数: 0 h-index: 0机构: Natl Inst Allergy & Infect Dis, Integrated Data Sci Sect, Res Technol Branch, NIH, Bethesda, MD USA NCI, Radiat Oncol Branch, 10 Ctr Dr MSC 1002,Bldg 10,B3B69B, Bethesda, MD 20892 USATofilon, Philip J.论文数: 0 引用数: 0 h-index: 0机构: NCI, Radiat Oncol Branch, 10 Ctr Dr MSC 1002,Bldg 10,B3B69B, Bethesda, MD 20892 USA NCI, Radiat Oncol Branch, 10 Ctr Dr MSC 1002,Bldg 10,B3B69B, Bethesda, MD 20892 USA