共 48 条
[1]
N-Benzyl-1-heteroaryl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamides as inhibitors of co-activator associated arginine methyltransferase 1 (CARM1)
[J].
Allan, Martin
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Manku, Sukhdev
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Therrien, Eric
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Nguyen, Natalie
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Styhler, Sylvia
;
Robert, Marie-France
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Goulet, Anne-Christine
;
Petschner, Andrea J.
;
Rahil, Gabi
;
MacLeod, A. Robert
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Deziel, Robert
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Besterman, Jeffrey M.
;
Nguyen, Hannah
;
Wahhab, Amal
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
2009, 19 (04)
:1218-1223

Allan, Martin
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Manku, Sukhdev
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Therrien, Eric
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Nguyen, Natalie
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Styhler, Sylvia
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Pharmacol & Cell Biol, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Robert, Marie-France
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Pharmacol & Cell Biol, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Goulet, Anne-Christine
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Pharmacol & Cell Biol, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Petschner, Andrea J.
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Lead Discovery, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Rahil, Gabi
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Lead Discovery, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

MacLeod, A. Robert
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Pharmacol & Cell Biol, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Deziel, Robert
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Besterman, Jeffrey M.
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Pharmacol & Cell Biol, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Nguyen, Hannah
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Pharmacol & Cell Biol, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada

Wahhab, Amal
论文数: 0 引用数: 0
h-index: 0
机构:
MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada MethylGene Inc, Dept Med Chem, Montreal, PQ H4S 2A1, Canada
[2]
Epigenetic protein families: a new frontier for drug discovery
[J].
Arrowsmith, Cheryl H.
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Bountra, Chas
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Fish, Paul V.
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Lee, Kevin
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Schapira, Matthieu
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NATURE REVIEWS DRUG DISCOVERY,
2012, 11 (05)
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Arrowsmith, Cheryl H.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada
Univ Toronto, Ontario Canc Inst, Toronto, ON M5G 1L7, Canada
Univ Toronto, Dept Med Biophys, Toronto, ON M5G 1L7, Canada Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Bountra, Chas
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Oxford, Nuffield Dept Clin Med, Struct Genom Consortium, Oxford OX3 7LD, England Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Fish, Paul V.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Ltd, Worldwide Med Chem, Sandwich CT13 9NJ, Kent, England Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

Lee, Kevin
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Immunoinflammat Ctr Excellence Drug Discovery, Epinova DPU, Stevenage SG1 2NY, Herts, England Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada

论文数: 引用数:
h-index:
机构:
[3]
Regulation of chromatin by histone modifications
[J].
Bannister, Andrew J.
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Kouzarides, Tony
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CELL RESEARCH,
2011, 21 (03)
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Bannister, Andrew J.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Cambridge, Gurdon Inst, Cambridge CB2 1QN, England
Univ Cambridge, Dept Pathol, Cambridge CB2 1QN, England Univ Cambridge, Gurdon Inst, Cambridge CB2 1QN, England

论文数: 引用数:
h-index:
机构:
[4]
Discovery of Peptidomimetic Ligands of EED as Allosteric Inhibitors of PRC2
[J].
Barnash, Kimberly D.
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The, Juliana
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Norris-Drouin, Jacqueline L.
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Cholensky, Stephanie H.
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Worley, Beau M.
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Li, Fengling
;
Stuckey, Jacob I.
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Brown, Peter J.
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Vedadi, Masoud
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Arrowsmith, Cheryl H.
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Frye, Stephen V.
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James, Lindsey I.
.
ACS COMBINATORIAL SCIENCE,
2017, 19 (03)
:161-172

Barnash, Kimberly D.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA

The, Juliana
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA

Norris-Drouin, Jacqueline L.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA

Cholensky, Stephanie H.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA

Worley, Beau M.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA

Li, Fengling
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA

Stuckey, Jacob I.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA

Brown, Peter J.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA

Vedadi, Masoud
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA

Arrowsmith, Cheryl H.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada
Univ Toronto, Princess Margaret Canc Ctr, Toronto, ON M5G 2M9, Canada
Univ Toronto, Dept Med Biophys, Toronto, ON M5G 2M9, Canada Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA

Frye, Stephen V.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA

James, Lindsey I.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA Univ N Carolina, UNC Eshelman Sch Pharm, Div Chem Biol & Med Chem, Ctr Integrat Chem Biol & Drug Discovery, Chapel Hill, NC 27599 USA
[5]
Pharmacologic Inhibition of the Menin-MLL Interaction Blocks Progression of MLL Leukemia In Vivo
[J].
Borkin, Dmitry
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He, Shihan
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Miao, Hongzhi
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Kempinska, Katarzyna
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Pollock, Jonathan
;
Chase, Jennifer
;
Purohit, Trupta
;
Malik, Bhavna
;
Zhao, Ting
;
Wang, Jingya
;
Wen, Bo
;
Zong, Hongliang
;
Jones, Morgan
;
Danet-Desnoyers, Gwenn
;
Guzman, Monica L.
;
Talpaz, Moshe
;
Bixby, Dale L.
;
Sun, Duxin
;
Hess, Jay L.
;
Muntean, Andrew G.
;
Maillard, Ivan
;
Cierpicki, Tomasz
;
Grembecka, Jolanta
.
CANCER CELL,
2015, 27 (04)
:589-602

Borkin, Dmitry
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

He, Shihan
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Miao, Hongzhi
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Kempinska, Katarzyna
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Pollock, Jonathan
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA
Univ Michigan, Grad Program Mol & Cellular Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Chase, Jennifer
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Inst Life Sci, Ctr Stem Cell Biol, Ann Arbor, MI 48109 USA
Univ Michigan, Grad Program Cellular & Mol Biol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

论文数: 引用数:
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Malik, Bhavna
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Zhao, Ting
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Wang, Jingya
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Wen, Bo
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Zong, Hongliang
论文数: 0 引用数: 0
h-index: 0
机构:
Cornell Univ, Weill Med Coll, Dept Med, New York, NY 10065 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

论文数: 引用数:
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机构:

Danet-Desnoyers, Gwenn
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Penn, Perelman Sch Med, Dept Med, Div Hematol Oncol, Philadelphia, PA 19104 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Guzman, Monica L.
论文数: 0 引用数: 0
h-index: 0
机构:
Cornell Univ, Weill Med Coll, Dept Med, New York, NY 10065 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Talpaz, Moshe
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Bixby, Dale L.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Sun, Duxin
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Coll Pharm, Dept Pharmaceut Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Hess, Jay L.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA
Indiana Univ, Sch Med, Indianapolis, IN 46202 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Muntean, Andrew G.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Maillard, Ivan
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Inst Life Sci, Ctr Stem Cell Biol, Ann Arbor, MI 48109 USA
Univ Michigan, Dept Internal Med, Div Hematol Oncol, Ann Arbor, MI 48109 USA
Univ Michigan, Dept Cell & Dev Biol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Cierpicki, Tomasz
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA

Grembecka, Jolanta
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Pathol, Ann Arbor, MI 48109 USA
[6]
Bromberg KD, 2017, NAT CHEM BIOL, V13, P317, DOI [10.1038/NCHEMBIO.2282, 10.1038/nchembio.2282]
[7]
Polycomb repressive complex 2 structure with inhibitor reveals a mechanism of activation and drug resistance
[J].
Brooun, Alexei
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Gajiwala, Ketan S.
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Deng, Ya-Li
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Liu, Wei
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Bolanos, Ben
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Bingham, Patrick
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He, You-Ai
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Diehl, Wade
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Grable, Nicole
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Kung, Pei-Pei
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Sutton, Scott
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Maegley, Karen A.
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Yu, Xiu
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Stewart, Al E.
.
NATURE COMMUNICATIONS,
2016, 7
:11384

Brooun, Alexei
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Gajiwala, Ketan S.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Deng, Ya-Li
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Liu, Wei
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Bolanos, Ben
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Bingham, Patrick
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Oncol Res Unit, Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

He, You-Ai
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Diehl, Wade
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Grable, Nicole
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Kung, Pei-Pei
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Sutton, Scott
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Maegley, Karen A.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Oncol Res Unit, Worldwide Res & Dev, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Yu, Xiu
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA

Stewart, Al E.
论文数: 0 引用数: 0
h-index: 0
机构:
Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA Pfizer Inc, Worldwide Res & Dev, Worldwide Med Chem, San Diego, CA 92121 USA
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Structure-Based Design of a Covalent Inhibitor of the SET Domain-Containing Protein 8 (SETD8) Lysine Methyltransferase
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Butler, Kyle V.
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Ma, Anqi
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Yu, Wenyu
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Li, Fengling
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Tempel, Wolfram
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Babault, Nicolas
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Pittella-Silva, Fabio
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Shao, Jason
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Wang, Junyi
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Luo, Minkui
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Vedadi, Masoud
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Brown, Peter J.
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Arrowsmith, Cheryl H.
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Jin, Jian
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JOURNAL OF MEDICINAL CHEMISTRY,
2016, 59 (21)
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Butler, Kyle V.
论文数: 0 引用数: 0
h-index: 0
机构:
Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA
Icahn Sch Med Mt Sinai, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Ma, Anqi
论文数: 0 引用数: 0
h-index: 0
机构:
Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA
Icahn Sch Med Mt Sinai, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Yu, Wenyu
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Li, Fengling
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Tempel, Wolfram
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Babault, Nicolas
论文数: 0 引用数: 0
h-index: 0
机构:
Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA
Icahn Sch Med Mt Sinai, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Pittella-Silva, Fabio
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Sloan Kettering Canc Ctr, Mol Pharmacol & Chem Program, New York, NY 10065 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Shao, Jason
论文数: 0 引用数: 0
h-index: 0
机构:
Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA
Icahn Sch Med Mt Sinai, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Wang, Junyi
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Sloan Kettering Canc Ctr, Mol Pharmacol & Chem Program, New York, NY 10065 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Luo, Minkui
论文数: 0 引用数: 0
h-index: 0
机构:
Mem Sloan Kettering Canc Ctr, Mol Pharmacol & Chem Program, New York, NY 10065 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Vedadi, Masoud
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada
Univ Toronto, Dept Pharmacol & Toxicol, Toronto, ON M5S 1A8, Canada Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Brown, Peter J.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Arrowsmith, Cheryl H.
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h-index: 0
机构:
Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada
Univ Toronto, Dept Pharmacol & Toxicol, Toronto, ON M5S 1A8, Canada Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA

Jin, Jian
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Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA
Icahn Sch Med Mt Sinai, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, New York, NY 10029 USA
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Scheufler, Clemens
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Klumpp, Martin
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Tiedt, Ralph
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Chen, Chao
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h-index: 0
机构:
Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Zhu, Hugh
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Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Stauffer, Frederic
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h-index: 0
机构:
Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Caravatti, Giorgio
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h-index: 0
机构:
Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Vollmer, Susanne
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Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Machauer, Rainer
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Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Holzer, Philipp
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机构:
Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Mobitz, Henrik
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Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Scheufler, Clemens
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Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Klumpp, Martin
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Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Tiedt, Ralph
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Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Beyer, Kim S.
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h-index: 0
机构:
Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Calkins, Keith
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h-index: 0
机构:
Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Guthy, Daniel
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h-index: 0
机构:
Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Kiffe, Michael
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h-index: 0
机构:
Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Zhang, Jeff
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Novartis Inst Biomed Res, Shanghai 201203, Peoples R China Novartis Inst Biomed Res, CH-4002 Basel, Switzerland

Gaul, Christoph
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h-index: 0
机构:
Novartis Inst Biomed Res, CH-4002 Basel, Switzerland Novartis Inst Biomed Res, CH-4002 Basel, Switzerland
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Copeland, Robert A.
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机构:
Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USA

Solomon, Michael E.
论文数: 0 引用数: 0
h-index: 0
机构:
Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USA

Richon, Victoria M.
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h-index: 0
机构:
Epizyme Inc, Cambridge, MA 02139 USA Epizyme Inc, Cambridge, MA 02139 USA