Unsymmetrical ureas. Synthetic methodologies and application in drug design

[1] Conversion of carbonimidodithioates into unsymmetrical di- and tri-substituted ureas including urea dipeptides [J]. TETRAHEDRON LETTERS, 1998, 39 (21) : 3609 - 3612

[2] Appelt Krzysztof, 1993, Perspectives in Drug Discovery and Design, V1, P23, DOI 10.1007/BF02171654

[3] A novel synthesis of disubstituted ureas using titanium(IV) isopropoxide and sodium borohydride [J]. TETRAHEDRON LETTERS, 1997, 38 (09) : 1531 - 1532

[4] A practical synthesis of cabergoline [J]. JOURNAL OF ORGANIC CHEMISTRY, 2002, 67 (20) : 7147 - 7150

[5] A new practical method for the synthesis of unsymmetrical ureas via high-pressure-promoted condensation of 2,2,2-trichloroethyl carbamates (Troc-carbamates) with amines [J]. TETRAHEDRON LETTERS, 2006, 47 (04) : 587 - 590

[6] SYNTHESIS OF N,N'-DISUBSTITUTED UREAS FROM CARBAMATES [J]. TETRAHEDRON LETTERS, 1988, 29 (21) : 2525 - 2526

[7] An efficient new protocol for the formation of unsymmetrical tri- and tetrasubstituted ureas [J]. TETRAHEDRON LETTERS, 1998, 39 (35) : 6267 - 6270

[8] REACTIONS OF AMINES .18. OXIDATIVE REARRANGEMENT OF AMIDES WITH LEAD-TETRAACETATE [J]. JOURNAL OF ORGANIC CHEMISTRY, 1975, 40 (24) : 3554 - 3561

[9] A simple desymmetrisation approach to unsymmetric N,N′-disubstituted cyclic ureas [J]. TETRAHEDRON LETTERS, 1999, 40 (39) : 7143 - 7146

[10] An efficient and convergent route towards water-soluble, chiral and amphiphilic macrocycles [J]. TETRAHEDRON LETTERS, 2001, 42 (15) : 2873 - 2875

[1] Conversion of carbonimidodithioates into unsymmetrical di- and tri-substituted ureas including urea dipeptides [J]. TETRAHEDRON LETTERS, 1998, 39 (21) : 3609 - 3612

[2] Appelt Krzysztof, 1993, Perspectives in Drug Discovery and Design, V1, P23, DOI 10.1007/BF02171654

[3] A novel synthesis of disubstituted ureas using titanium(IV) isopropoxide and sodium borohydride [J]. TETRAHEDRON LETTERS, 1997, 38 (09) : 1531 - 1532

[4] A practical synthesis of cabergoline [J]. JOURNAL OF ORGANIC CHEMISTRY, 2002, 67 (20) : 7147 - 7150

[5] A new practical method for the synthesis of unsymmetrical ureas via high-pressure-promoted condensation of 2,2,2-trichloroethyl carbamates (Troc-carbamates) with amines [J]. TETRAHEDRON LETTERS, 2006, 47 (04) : 587 - 590

[6] SYNTHESIS OF N,N'-DISUBSTITUTED UREAS FROM CARBAMATES [J]. TETRAHEDRON LETTERS, 1988, 29 (21) : 2525 - 2526

[7] An efficient new protocol for the formation of unsymmetrical tri- and tetrasubstituted ureas [J]. TETRAHEDRON LETTERS, 1998, 39 (35) : 6267 - 6270

[8] REACTIONS OF AMINES .18. OXIDATIVE REARRANGEMENT OF AMIDES WITH LEAD-TETRAACETATE [J]. JOURNAL OF ORGANIC CHEMISTRY, 1975, 40 (24) : 3554 - 3561

[9] A simple desymmetrisation approach to unsymmetric N,N′-disubstituted cyclic ureas [J]. TETRAHEDRON LETTERS, 1999, 40 (39) : 7143 - 7146

[10] An efficient and convergent route towards water-soluble, chiral and amphiphilic macrocycles [J]. TETRAHEDRON LETTERS, 2001, 42 (15) : 2873 - 2875