An Efficient Protein System for Screening Specific MdmX and Mdm2 Inhibitors

被引:0
|
作者
Chen, Rong [1 ]
Zhou, Jingjing [1 ]
Qin, Lingyun [1 ]
Su, Zhengding [1 ]
机构
[1] Hubei Univ TEchnol, Wuhan, Peoples R China
关键词
D O I
10.1016/j.bpj.2016.11.2680
中图分类号
Q6 [生物物理学];
学科分类号
071011 ;
摘要
2438-Pos
引用
收藏
页码:495A / 495A
页数:1
相关论文
共 50 条
  • [11] The MDM2 RING Domain and Central Acidic Domain Play Distinct Roles in MDM2 Protein Homodimerization and MDM2-MDMX Protein Heterodimerization
    Leslie, Patrick L.
    Ke, Hengming
    Zhang, Yanping
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2015, 290 (20) : 12941 - 12950
  • [12] MDM2 promotes ubiquitination and degradation of MDMX
    Pan, Y
    Chen, JD
    MOLECULAR AND CELLULAR BIOLOGY, 2003, 23 (15) : 5113 - 5121
  • [13] Role of Mdm2 and Mdmx in DNA repair
    Eischen, Christine M.
    JOURNAL OF MOLECULAR CELL BIOLOGY, 2017, 9 (01) : 69 - 73
  • [14] DISRUPTION OF P53/MDM2/MDMX PROTEIN-PROTEIN INTERACTIONS
    Topper, M.
    Zhou, M.
    Anderson, L.
    McLaughlin, M.
    BIOPOLYMERS, 2009, 92 (04) : 332 - 332
  • [15] Mdm2 and MdmX inhibitors for the treatment of cancer: a patent review (2011-present)
    Zak, Krzysztof
    Pecak, Aleksandra
    Rys, Barbara
    Wladyka, Benedykt
    Doemling, Alexander
    Weber, Lutz
    Holak, Tad A.
    Dubin, Grzegorz
    EXPERT OPINION ON THERAPEUTIC PATENTS, 2013, 23 (04) : 425 - 448
  • [16] Ligand Binding Mode Prediction by Docking: Mdm2/Mdmx Inhibitors as a Case Study
    Bharatham, Nagakumar
    Bharatham, Kavitha
    Shelat, Anang A.
    Bashford, Donald
    JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2014, 54 (02) : 648 - 659
  • [17] Searching for novel MDM2/MDMX dual inhibitors through a drug repurposing approach
    Li, Keting
    Hu, Wenshu
    Wang, Yingjie
    Chen, Wenxing
    Wen, Hongmei
    Liu, Jian
    Li, Wei
    Wang, Bo
    JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2024, 39 (01)
  • [18] MdmX inhibits ARF mediated Mdm2 sumoylation
    Ghosh, M
    Weghorst, K
    Berberich, SJ
    CELL CYCLE, 2005, 4 (04) : 604 - 608
  • [19] MdmX Protein Is Essential for Mdm2 Protein-mediated p53 Polyubiquitination
    Wang, Xinjiang
    Wang, Junru
    Jiang, Xuejun
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2011, 286 (27) : 23725 - 23734
  • [20] Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: Identification of novel peptidic inhibitors
    Noguchi, Taro
    Oishi, Shinya
    Honda, Kaori
    Kondoh, Yasumitsu
    Saito, Tamio
    Kubo, Tatsuhiko
    Kaneda, Masato
    Ohno, Hiroaki
    Osada, Hiroyuki
    Fujii, Nobutaka
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (13) : 3802 - 3805