SYNTHESIS OF TWO ISOTOPICALLY LABELED VERSIONS OF AURORA A KINASE INHIBITOR

被引:0
|
作者
Li, Yuexian [1 ]
Prakash, Shimoga R. [1 ]
机构
[1] Takeda Oncol Co, Millennium Pharmaceut Inc, Isotope Chem Grp, Dept Drug Metab & Pharmacokinet, Cambridge, MA 02139 USA
来源
关键词
C-14]-sodium 4-[[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-2-methoxy benzoate; (CD3)-C-13,N-15(2)]-sodium 4-[[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-2-methoxy benzoate; SMALL-MOLECULE INHIBITOR; IKK INHIBITOR; MLN8054; C-14; H-3;
D O I
暂无
中图分类号
Q5 [生物化学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:448 / 450
页数:3
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