SYNTHESIS CHARACTERIZATION AND BIOLOGICAL EVALUATION OF NOVEL OF (1E)-1-((9-((4,5-DIHYDRO-5-THIOXO-1,3,4-OXADIAZOL-2-YL)METHYL)-9H-CARBAZOL-6-YL)METHYLENE)THIOSEMICARBAZIDE BEARING PHENYL THIAZOLE

被引：0

作者：

Krishna, S. Murali ^{[1
]}

Raveendra, M. ^{[1
]}

机构：

[1] Rajiv Gandhi Univ Knowledge Technol, DrAPJ Abdulkalam IIT ONGOLE, Biol E Ltd Co, Hyderabad, Telangana, India

来源：

HETEROCYCLIC LETTERS | 2019年 / 9卷 / 04期

关键词：

Antibacterial activity; Antifungal activity; carbazole; thiazole; CARBAZOLE; ALKALOIDS; INDOLE;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The article is aimed to synthesize, characterize and screening the biological activity of (1E)-1-((9-((4,5-dihy dro-5-thi oxo-1,3,4-oxadi azol-2-yl)methyl)-9H-carb azol-6-yl)methylene)thi osemicarbazi de bearing phenyl thiazole The structure of these newly synthesized compounds were characterised by H-1 NMR, (CNMR)-C-13 ,Mass ,IR, and elemental analysis. The antimicriobial activity of the novel compounds was screened by agar disc diffusion method

引用

页码：481 / 486

页数：6

共 50 条

[21] DESIGN AND SYNTHESIS OF NOVEL 2-(4-((5-PHENYL-1, 3, 4-OXADIAZOL-2-YL)METHOXY)SUBSTITUTEDPHENYL)-1H-BENZO [de]ISOQUINOLINE-1, 3(2H)-DIONE DERIVATIVE AS ANTIBACTERIAL AND ANTIFUNGAL AGENTS [J].

Sirgamalla, Rambabu ;

Kommakula, Ashok ;

Sakram, Boda ;

Kumar, B. Sathish ;

Lakshmi, P. V. Anantha .

HETEROCYCLIC LETTERS, 2018, 8 (04) :831-842

[22] Synthesis, Characterization, and Biological Studies of Organometallic Compounds of Re(I) with 2-(5-(4-Nitrophenyl)-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzo[d]thiazole Based Derivatives [J].

Padariya, Aelvish D. ;

Savaliya, Nirbhay K. ;

Parekh, Hitesh M. ;

Bhatt, Bhupesh S. ;

Bhatt, Vaibhav D. ;

Patel, Mohan N. .

CHEMISTRYSELECT, 2025, 10 (21)

[23] Synthesis, Characterization and Antimicrobial Evaluation of Novel (E)-N'-(4-(1-((3,4-dimethoxypyridin-2-yl)methyl)-1H-1,2,3-triazol-4-yl)benzylidene)benzohydrazide Derivatives [J].

Saidugari, Swamy ;

Vadali, Lakshmana Rao ;

Vidya, K. ;

Ram, B. .

ORIENTAL JOURNAL OF CHEMISTRY, 2016, 32 (04) :2155-2161

[24] Synthesis and Biological Activities of Novel N-(5-Alkyl-1,3,4-thiadiazol-2-yl)-1-[(heteroaryl)methyl]-5-methyl-1H-1,2,3-triazole-4-carboxamides [J].

Chen, Xiaobao ;

Shi, Deqing .

CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2009, 29 (07) :1096-1099

[25] Synthesis, characterization, biological evaluation and docking studies of novel 5-(2-methyl-1,8-naphthyridin-3-yl)-1,3,4-oxadiazol-2-amine and some of its derivatives using symmetrical anhydrides [J].

Parangi, Ravi Kumar ;

Domala, Ramesh .

RESULTS IN CHEMISTRY, 2023, 5

[26] Synthesis and antimicrobial evaluation of 1-(benzofuran-2-yl)-4-nitro-3-arylbutan-1-ones and 3-(benzofuran-2-yl)-4,5-dihydro-5-aryl-1-[4-(aryl)-1, 3-thiazol-2-yl]-1H-pyrazoles [J].

Abdel-Wahab, Bakr F. ;

Abdel-Aziz, Hatem A. ;

Ahmed, Essam M. .

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2009, 44 (06) :2632-2635

[27] SYNTHESIS AND CHARACTERIZATION OF (Z)-N-(1-[2-{3-[(DIMETHYLAMINO)METHYL)]-2-METHOXYPHENYL}-5-(PY RIDIN-4-YL)-1,3,4-OXADIAZOL-3(2H)-YL]ETHYLIDENE) BENZENAMINE DERIVATIVES AS POTENT ANTIFUNGAL AGENTS [J].

Malhotra, Manav ;

Hans, Pankhuri ;

Sharma, Sagun ;

Deep, Aakash ;

Phogat, Priyanka .

ACTA POLONIAE PHARMACEUTICA, 2012, 69 (03) :433-438

[28] Synthesis, in vitro and in silico studies of novel potent urease inhibitors: N-[4-({5-[(3-Un/ubstituted-anilino-3-oxopropyl) sulfanyl]-1,3,4-oxadiazol-2-yl} methyl)-1,3-thiazol-2-yl] benzamides [J].

Abbasi, Muhammad Athar ;

Hassan, Mubashir ;

Aziz-ur-Rehman ;

Siddiqui, Sabahat Zahra ;

Raza, Hussain ;

Shah, Syed Adnan Ali ;

Seo, Sung-Yum .

BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 26 (13) :3791-3804

[29] Synthesis and antimicrobial screening of novel 9-{2-[(1H-1,2,3-triazol-4-yl)methoxy]phenyl}-3,3,6,6-tetramethyl-3,4,5,6,7,9-hexahydro-1H-xanthene-1,8(2H)-dione derivatives [J].

A. Kishore Kumar ;

V. Sunitha ;

B. Shankar ;

T. Murali Krishna ;

Ch. Abraham Lincoln ;

P. Jalapathi .

Russian Journal of General Chemistry, 2017, 87 :2011-2020

[30] Synthesis and antimicrobial screening of novel 9-{2-[(1H-1,2,3-triazol-4-yl)methoxy]phenyl}-3,3,6,6-tetramethyl-3,4,5,6,7,9-hexahydro-1H-xanthene-1,8(2H)-dione derivatives [J].

Kumar, A. Kishore ;

Sunitha, V. ;

Shankar, B. ;

Krishna, T. Murali ;

Lincoln, Ch. Abraham ;

Jalapathi, P. .

RUSSIAN JOURNAL OF GENERAL CHEMISTRY, 2017, 87 (09) :2011-2020

← 1 2 3 4 5 →