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- [21] Structure-Guided Design, Synthesis, and Antivirulence Assessment of Covalent Staphylococcus aureus Sortase A InhibitorsJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (02) : 1127 - 1146Yue, Chuan论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Ctr Chem Biol, State Key Lab Drug Res, Shanghai 201203, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaYuan, Ziqi论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Ctr Chem Biol, State Key Lab Drug Res, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaXu, Guobin论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Ctr Chem Biol, State Key Lab Drug Res, Shanghai 201203, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Ctr Chem Biol, State Key Lab Drug Res, Shanghai 201203, Peoples R China China Pharmaceut Univ, Sch Pharm, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 210009, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaGuan, Xiang-Na论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Ctr Chem Biol, State Key Lab Drug Res, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaWei, Bingyan论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Ctr Chem Biol, State Key Lab Drug Res, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China Univ Chinese Acad Sci, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, Hangzhou 310024, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaYao, Hequan论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Pharm, State Key Lab Nat Med, Nanjing 210009, Peoples R China China Pharmaceut Univ, Sch Pharm, Dept Med Chem, Nanjing 210009, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaYang, Cai-Guang论文数: 0 引用数: 0 h-index: 0机构: Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China Chinese Acad Sci, Shanghai Inst Mat Med, Ctr Chem Biol, State Key Lab Drug Res, Shanghai 201203, Peoples R China Univ Chinese Acad Sci, Beijing 100049, Peoples R China Univ Chinese Acad Sci, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, Hangzhou 310024, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R ChinaZhang, Tao论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Shanghai Inst Mat Med, Ctr Chem Biol, State Key Lab Drug Res, Shanghai 201203, Peoples R China Nanjing Univ Chinese Med, Sch Chinese Mat Med, Nanjing 210023, Peoples R China
- [22] Polar protein-ligand interactions: Statistical significance and use in structure-guided drug designABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 255Kuhn, Bernd论文数: 0 引用数: 0 h-index: 0机构: F Hoffmann La Roche, Basel, Switzerland F Hoffmann La Roche, Basel, Switzerland
- [23] Crystal Structure-Guided Design of Bisubstrate Inhibitors and Photoluminescent Probes for Protein Kinases of the PIM FamilyMOLECULES, 2021, 26 (14):Nonga, Olivier E.论文数: 0 引用数: 0 h-index: 0机构: Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, Estonia Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, EstoniaLavogina, Darja论文数: 0 引用数: 0 h-index: 0机构: Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, Estonia Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, Estonia论文数: 引用数: h-index:机构:Kestav, Katrin论文数: 0 引用数: 0 h-index: 0机构: Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, Estonia Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, Estonia论文数: 引用数: h-index:机构:Dixon-Clarke, Sarah E.论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Ctr Med Discovery, Old Rd Campus,Roosevelt Dr, Oxford OX3 7DQ, England Dana Farber Canc Inst, Dept Canc Biol, 450 Brookline Ave, Boston, MA 02215 USA Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, EstoniaBullock, Alex N.论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Ctr Med Discovery, Old Rd Campus,Roosevelt Dr, Oxford OX3 7DQ, England Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, EstoniaKopanchuk, Sergei论文数: 0 引用数: 0 h-index: 0机构: Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, Estonia Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, Estonia论文数: 引用数: h-index:机构:Ekambaram, Ramesh论文数: 0 引用数: 0 h-index: 0机构: Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, Estonia Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, EstoniaViht, Kaido论文数: 0 引用数: 0 h-index: 0机构: Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, Estonia Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, EstoniaKnapp, Stefan论文数: 0 引用数: 0 h-index: 0机构: Goethe Univ Frankfurt Main, Inst Pharmazeut Chem, Max von Laue Str 9, D-60438 Frankfurt, Germany Goethe Univ Frankfurt, Buchmann Inst Life Sci, Struct Genom Consortium SGC, Max von Laue Str 15, D-60438 Frankfurt, Germany Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, EstoniaUri, Asko论文数: 0 引用数: 0 h-index: 0机构: Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, Estonia Univ Tartu, Inst Chem, 14A Ravila St, EE-50411 Tartu, Estonia
- [24] Identification and structure-guided enzyme engineering of an extremophilic protein phosphataseFASEB JOURNAL, 2020, 34Chen, Tiantian论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Lexington, KY 40506 USA Univ Kentucky, Lexington, KY 40506 USAKooi, Carl论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Lexington, KY 40506 USA Univ Kentucky, Lexington, KY 40506 USAAnwar, Humza论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Lexington, KY 40506 USA Univ Kentucky, Lexington, KY 40506 USASharma, Savita论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Lexington, KY 40506 USA Univ Kentucky, Lexington, KY 40506 USA论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Kooi, Craig论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Lexington, KY 40506 USA Univ Kentucky, Lexington, KY 40506 USA
- [25] Structure-guided discovery of protein and glycan components in native mastigonemesCELL, 2024, 187 (07) : 1733 - 1744.e12Huang, Junhao论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R China Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R ChinaTao, Hui论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Life Sci, Tsinghua Peking Joint Ctr Life Sci, MOE Key Lab Prot Sci, Beijing 100084, Peoples R China Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R ChinaChen, Jikun论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Life Sci, Tsinghua Peking Joint Ctr Life Sci, MOE Key Lab Prot Sci, Beijing 100084, Peoples R China Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R ChinaShen, Yang论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R China Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R ChinaLei, Jianlin论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R China Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R ChinaPan, Junmin论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Life Sci, Tsinghua Peking Joint Ctr Life Sci, MOE Key Lab Prot Sci, Beijing 100084, Peoples R China Qingdao Natl Lab Marine Sci & Technol, Lab Marine Biol & Biotechnol, Qingdao, Shandong, Peoples R China Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R ChinaYan, Chuangye论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R China Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R ChinaYan, Nieng论文数: 0 引用数: 0 h-index: 0机构: Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R China Shenzhen Med Acad Res & Translat Smart, Inst Bioarchitecture & Biointeract IBABI, Shenzhen 518107, Guangdong, Peoples R China Tsinghua Univ, Sch Life Sci, State Key Lab Membrane Biol, Beijing Frontier Res Ctr Biol Struct,Tsinghua Pek, Beijing 100084, Peoples R China
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- [27] Structure-guided design of antibacterials that allosterically inhibit DNA gyraseBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 29 (11) : 1407 - 1412Thalji, Reema K.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline, Collegeville, PA 19426 USARaha, Kaushik论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline, Collegeville, PA 19426 USAAndreotti, Daniele论文数: 0 引用数: 0 h-index: 0机构: EVOTEC Ctr Drug Discovery & Dev, I-37135 Verona, Italy GlaxoSmithKline, Collegeville, PA 19426 USAChecchia, Anna论文数: 0 引用数: 0 h-index: 0机构: EVOTEC Ctr Drug Discovery & Dev, I-37135 Verona, Italy GlaxoSmithKline, Collegeville, PA 19426 USACui, Haifeng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline, Collegeville, PA 19426 USAMeneghelli, Giovanni论文数: 0 引用数: 0 h-index: 0机构: EVOTEC Ctr Drug Discovery & Dev, I-37135 Verona, Italy FIS, I-36075 Vicenza, Italy GlaxoSmithKline, Collegeville, PA 19426 USAProfeta, Roberto论文数: 0 引用数: 0 h-index: 0机构: EVOTEC Ctr Drug Discovery & Dev, I-37135 Verona, Italy FIS, I-36075 Vicenza, Italy GlaxoSmithKline, Collegeville, PA 19426 USATonelli, Federica论文数: 0 引用数: 0 h-index: 0机构: EVOTEC Ctr Drug Discovery & Dev, I-37135 Verona, Italy GlaxoSmithKline, Collegeville, PA 19426 USATommasi, Simona论文数: 0 引用数: 0 h-index: 0机构: EVOTEC Ctr Drug Discovery & Dev, I-37135 Verona, Italy FIS, I-36075 Vicenza, Italy GlaxoSmithKline, Collegeville, PA 19426 USABakshi, Tania论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline, Collegeville, PA 19426 USADonovan, Brian T.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline, Collegeville, PA 19426 USAHowells, Alison论文数: 0 引用数: 0 h-index: 0机构: Inspiralis Ltd, Innovat Ctr, Norwich NR4 7GJ, Norfolk, England GlaxoSmithKline, Collegeville, PA 19426 USAJain, Shruti论文数: 0 引用数: 0 h-index: 0机构: Inspiralis Ltd, Innovat Ctr, Norwich NR4 7GJ, Norfolk, England GlaxoSmithKline, Collegeville, PA 19426 USANixon, Christopher论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline, Collegeville, PA 19426 USAQuinque, Geoffrey论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline, Collegeville, PA 19426 USAMcCloskey, Lynn论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline, Collegeville, PA 19426 USABax, Benjamin D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Stevenage SG1 2NYH, Herts, England Cardiff Univ, Med Discovery Inst, Main Bldg,Pk Pl, Cardiff CF10 3AT, S Glam, Wales GlaxoSmithKline, Collegeville, PA 19426 USANeu, Margarete论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Stevenage SG1 2NYH, Herts, England GlaxoSmithKline, Collegeville, PA 19426 USAChan, Pan F.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline, Collegeville, PA 19426 USAStavenger, Robert A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline, Collegeville, PA 19426 USA
- [28] Structure-Guided Design of Potent Diazobenzene Inhibitors for the BET BromodomainsJOURNAL OF MEDICINAL CHEMISTRY, 2013, 56 (22) : 9251 - 9264Zhang, Guangtao论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USAPlotnikov, Alexander N.论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USARusinova, Elena论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USAShen, Tong论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USAMorohashi, Keita论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USAJoshua, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USAZeng, Lei论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USAMujtaba, Shiraz论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USAOhlmeyer, Michael论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USAZhou, Ming-Ming论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Struct & Chem Biol, New York, NY 10029 USA
- [29] Structure-guided design of a high-affinity ligand for a riboswitchRNA, 2019, 25 (04) : 423 - 430Huang, Lin论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Canc Res UK Nucle Acid Struct Res Grp, MSI WTB Complex, Dundee DD1 5EH, Scotland Univ Dundee, Canc Res UK Nucle Acid Struct Res Grp, MSI WTB Complex, Dundee DD1 5EH, ScotlandWang, Jia论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Canc Res UK Nucle Acid Struct Res Grp, MSI WTB Complex, Dundee DD1 5EH, Scotland Univ Dundee, Canc Res UK Nucle Acid Struct Res Grp, MSI WTB Complex, Dundee DD1 5EH, ScotlandWilson, Timothy J.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Canc Res UK Nucle Acid Struct Res Grp, MSI WTB Complex, Dundee DD1 5EH, Scotland Univ Dundee, Canc Res UK Nucle Acid Struct Res Grp, MSI WTB Complex, Dundee DD1 5EH, ScotlandLilley, David M. J.论文数: 0 引用数: 0 h-index: 0机构: Univ Dundee, Canc Res UK Nucle Acid Struct Res Grp, MSI WTB Complex, Dundee DD1 5EH, Scotland Univ Dundee, Canc Res UK Nucle Acid Struct Res Grp, MSI WTB Complex, Dundee DD1 5EH, Scotland
- [30] Structure-guided design of a potent Clostridiodes difficile toxin A inhibitorFRONTIERS IN MICROBIOLOGY, 2023, 14Hussack, Greg论文数: 0 引用数: 0 h-index: 0机构: Natl Res Council Canada, Human Hlth Therapeut Res Ctr, Life Sci Div, Ottawa, ON, Canada Natl Res Council Canada, Human Hlth Therapeut Res Ctr, Life Sci Div, Ottawa, ON, CanadaRossotti, Martin A.论文数: 0 引用数: 0 h-index: 0机构: Natl Res Council Canada, Human Hlth Therapeut Res Ctr, Life Sci Div, Ottawa, ON, Canada Natl Res Council Canada, Human Hlth Therapeut Res Ctr, Life Sci Div, Ottawa, ON, Canadavan Faassen, Henk论文数: 0 引用数: 0 h-index: 0机构: Natl Res Council Canada, Human Hlth Therapeut Res Ctr, Life Sci Div, Ottawa, ON, Canada Natl Res Council Canada, Human Hlth Therapeut Res Ctr, Life Sci Div, Ottawa, ON, CanadaMurase, Tomohiko论文数: 0 引用数: 0 h-index: 0机构: Univ Calgary, Dept Biol Sci, Calgary, AB, Canada Natl Res Council Canada, Human Hlth Therapeut Res Ctr, Life Sci Div, Ottawa, ON, CanadaEugenio, Luiz论文数: 0 引用数: 0 h-index: 0机构: Univ Calgary, Dept Biol Sci, Calgary, AB, Canada Natl Res Council Canada, Human Hlth Therapeut Res Ctr, Life Sci Div, Ottawa, ON, CanadaSchrag, Joseph D.论文数: 0 引用数: 0 h-index: 0机构: Natl Res Council Canada, Human Hlth Therapeut Res Ctr, Life Sci Div, Montreal, PQ, Canada Natl Res Council Canada, Human Hlth Therapeut Res Ctr, Life Sci Div, Ottawa, ON, CanadaNg, Kenneth K. -S.论文数: 0 引用数: 0 h-index: 0机构: Univ Calgary, Dept Biol Sci, Calgary, AB, Canada Univ Windsor, Dept Chem & Biochem, Windsor, ON, Canada Natl Res Council Canada, Human Hlth Therapeut Res Ctr, Life Sci Div, Ottawa, ON, Canada论文数: 引用数: h-index:机构: