Microwave-promoted, solvent-free, three-component coupling of aldehyde, alkyne, and amine catalyzed by AgNO3

被引：12

作者：

He, Tingting ^{[1
]}

Zha, Zhenggen ^{[1
]}

Pan, Chongfeng ^{[1
]}

Wang, Zhiyong ^{[1
]}

机构：

[1] Univ Sci & Technol China, Dept Chem, Natl Lab Phys Sci Microscale, Hefei 230026, Peoples R China

来源：

SYNTHETIC COMMUNICATIONS | 2007年 / 37卷 / 4-6期

基金：

中国国家自然科学基金;

关键词：

microwave; propargylamine; silver catalyst; solvent free; three-component coupling;

D O I：

10.1080/00397910601131320

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient three-component coupling reaction of alkyne, aldehyde, and amine was carried out in one pot smoothly under the catalysis of AgNO3 and microwave irradiation. The scope of reaction substrates was extended. Moreover, the reaction can be performed under solvent-free condition, affording propargylarnine derivatives with high yields.

引用

页码：849 / 858

页数：10

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