Microwave assisted improved synthesis of 6-formylpterin and other heterocyclic mono- and di-aldehydes

被引：26

作者：

Goswami, S ^{[1
]}

Adak, AK ^{[1
]}

机构：

[1] Deemed Univ, Bengal Engn Coll, Dept Chem, Howrah 711103, W Bengal, India

来源：

SYNTHETIC COMMUNICATIONS | 2003年 / 33卷 / 03期

关键词：

selenium dioxide; 6-formylpterin; heterocyclic aldehyde; microwave;

D O I：

10.1081/SCC-120015779

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

2-Pivaloylamino-6-formylpterin (1a) and a series of other important heterocyclic aldehydes (2a, 3a, 4a, 6a, and 7a) have been synthesized in good yield by microwave assisted selenium dioxide oxidation. Interestingly, 2-methylpyrazine gives 2-pyrazinecarboxylic acid (5a) under the similar condition.

引用

页码：475 / 480

页数：6

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