Efficacy and Safety of ABT-126 in Subjects with Mild-to-Moderate Alzheimer's Disease on Stable Doses of Acetylcholinesterase Inhibitors: A Randomized, Double-Blind, Placebo-Controlled Study

被引:28
作者
Florian, Hana [1 ]
Meier, Andreas [1 ,5 ]
Gauthier, Serge [2 ]
Lipschitz, Stanley [3 ]
Lin, Yunzhi [1 ,6 ]
Tang, Qi [1 ]
Othman, Ahmed A. [1 ,4 ]
Robieson, Weining Z. [1 ]
Gault, Laura M. [1 ]
机构
[1] AbbVie Inc, 1 North Waukegan Rd,Bldg AP31-1, N Chicago, IL 60064 USA
[2] McGill Univ, Res Ctr Studies Aging, Montreal, PQ, Canada
[3] Dr Stanley Lipschitz Clin, Rosebank, Johannesburg, South Africa
[4] Cairo Univ, Fac Pharm, Dept Pharmaceut, Cairo, Egypt
[5] Pfizer Inc, Cambridge, MA USA
[6] Takeda Pharmaceut USA Inc, Deerfield, IL USA
关键词
ABT-126; Acetylcholinesterase inhibitors; alzheimer's disease; dementia; nicotinic acetylcholine receptors; NICOTINIC PARTIAL AGONIST; ANTIPSYCHOTIC EFFICACY; RECEPTOR; SCHIZOPHRENIA; COGNITION; DEFICITS; EVP-6124; MEMORY; GTS-21; TRIAL;
D O I
10.3233/JAD-150978
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
Background: ABT-126 is a potent, selective alpha 7 nicotinic acetylcholine receptor agonist with putative procognitive effects as a monotherapy in treating Alzheimer's disease (AD). Objective: This randomized, double-blind, placebo-controlled multicenter study (NCT01549834) investigated the efficacy and safety of ABT-126 in subjects with mild-to-moderate AD who were taking stable doses of acetylcholinesterase inhibitors (AChEIs). Methods: Subjects received 25mg ABT-126 (n = 143), 75 mg ABT-126 (n = 145), or placebo (n = 146) once daily for 24 weeks. Subjects who completed the 24-week double-blind study were eligible to enroll in a 28-week open-label extension study (NCT01690195) and received 75mg ABT-126 daily. The primary efficacy endpoint was the change from baseline to week 24 in the 11-item total score of the Alzheimer's Disease Assessment Scale-Cognitive Subscale (ADAS-Cog). Results: Neither dose of ABT-126 demonstrated significant improvement compared with placebo in the primary efficacy endpoint. However, 25 mg ABT-126 demonstrated significant improvement compared with placebo in ADAS-Cog scores at week 4 (least squares mean difference, -1.21; standard error, 0.51; p < 0.010, one-sided); 75 mg ABT-126 did not demonstrate significant improvements in ADAS-Cog scores compared with placebo at any time point. A treatment effect was not observed for any secondary efficacy measures of cognition, function, or global improvement. ABT-126 was generally well tolerated; the most common adverse events were agitation, constipation, diarrhea, fall, and headache. Conclusions: Overall, the efficacy profile of ABT-126 did not warrant further development as add-on therapy to AChEIs to treat mild-to-moderate AD.
引用
收藏
页码:1237 / 1247
页数:11
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