Microwave assisted one-pot synthesis of linear and angular furo chromanone scaffolds and their in vitro antimicrobial activity

被引：1

作者：

Venkataramana, R. ^{[1
]}

Reddy, Ch. Venkata Ramana ^{[2
]}

Ashok, D. ^{[3
]}

Nagaraju, N. ^{[4
]}

机构：

[1] IDA, Sebond Sci, Hyderabad 500076, Telangana, India

[2] Jawaharlal Nehru Technol Univ, Dept Chem, Hyderabad 500085, Telangana, India

[3] Osmania Univ, Dept Chem, Hyderabad 500007, Telangana, India

[4] Osmania Univ, Dept Microbiol, Hyderabad 500007, Telangana, India

来源：

RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2017年 / 87卷 / 04期

关键词：

furochromanone; aliphaticaldehydes; microwave irradiation; antimicrobial activity; CONDENSATION;

D O I：

10.1134/S1070363217040302

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A new series of linear and angular alkyl substituted furochromanone derivatives have been synthesized in one pot microwave irradiation assisted process from ortho-hydroxy acetyl (linear and angular) benzofurans and aliphatic aldehydes in the presence of pyrrolidine. Various alkyl substituted furochromanones were synthesized with high yields. The in vitro antimicrobial activity of the products was tested. The structures of the compound have been elucidated on the basis of elemental analysis, IR, H-1 and C-13 NMR, and MS spectral data.

引用

页码：850 / 856

页数：7

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