Cyclisation of tryptamine enaminones to functionalised tetrahydro-β-carbolines induced by [bis(trifluoroacetoxy)iodo]benzene

被引：16

作者：

Papadopoulou, D ^{[1
]}

Papoutsis, I ^{[1
]}

Spyroudis, S ^{[1
]}

Varvoglis, A ^{[1
]}

机构：

[1] Univ Thessaloniki, Dept Chem, Organ Chem Lab, GR-54006 Thessaloniki, Greece

来源：

TETRAHEDRON LETTERS | 1998年 / 39卷 / 18期

关键词：

D O I：

10.1016/S0040-4039(98)00319-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The reaction of enamino carbonyl derivatives of tryptamine with [bis(trifluoroacetoxy)iodo]benzene provides an easy route to 1,1-bis-functionalised-N-trifluoroacetylated-beta-carbolines. The reaction proceeds through Pictet-Spengler-type cyclisation, trifluoroacetylation and oxidation steps. (C) 1998 Elsevier Science Ltd. All rights reserved.

引用

页码：2865 / 2866

页数：2