Use of 3,5-disubstituted 1,2,4-triazoles for the synthesis of peptidomimetics

被引：10

作者：

Cesar, J ^{[1
]}

Sollner, M ^{[1
]}

机构：

[1] Univ Ljubljana, Fac Pharm, Ljubljana 1000, Slovenia

来源：

SYNTHETIC COMMUNICATIONS | 2000年 / 30卷 / 22期

关键词：

D O I：

10.1080/00397910008087031

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of 3-acylaminoalkyl-5-alkyloxycarbonyl-1,2,4-triazoles, designed as RGD peptidomimetics, is described and the reactivity of 1,2,4-triazoles under conditions of peptide chemistry is discussed.

引用

页码：4147 / 4158

页数：12

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