Advances in the Synthesis of Nitrogen Zole s-Triazine Compounds

被引：1
|
作者：
Wang, Tao [1 ]
Xie, Zhongpao [1 ]
Zeng, Ming [1 ]
Cui, Dongmei [1 ]
机构：
[1] Zhejiang Univ Technol, Coll Pharmaceut Sci, Hangzhou 310014, Zhejiang, Peoples R China
来源：
CHINESE JOURNAL OF ORGANIC CHEMISTRY | 2018年 / 38卷 / 05期
关键词：
nitrogen zole; s-triazine; tetrazolo-s-triazine; triazolo-s-triazine; diazolo-s-triazine; ANTI-THYMIDINE PHOSPHORYLASE; MICROWAVE-ASSISTED SYNTHESIS; STRUCTURE-BASED DESIGN; CONVENIENT SYNTHESIS; TRANSLOCATIVE REARRANGEMENTS; CONTAINING HETEROCYCLES; BIOLOGICAL-ACTIVITY; POTENT INHIBITORS; ADENOSINE A(2A); C-NUCLEOSIDE;
D O I：
10.6023/cjoc201711046
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Nitrogen zole s-triazine derivatives display several biological activities such as antiproliferative, antioxidant, antiviral, antitumor and so on. Accordingly, much effort has been made towards the development of diverse synthetic methods for nitrogen zole s-triazines. The advancements in synthesis of nitrogen zole s-triazine compounds are summarized, including tetrazolo-s-triazines, triazolo-s-triazines and diazolo-s-triazines. At last the disadvantages of these synthetic methods are discussed and prospected to the future development.
引用
收藏
页码：983 / 998
页数：16
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