Synthesis of constrained α-amino acid derivatives via Diels-Alder approach

被引:61
|
作者
Kotha, S [1 ]
Brahmachary, E [1 ]
Sreenivasachary, N [1 ]
机构
[1] Indian Inst Technol, Dept Chem, Bombay 400076, Maharashtra, India
关键词
alkynes; amino acids; Diels-Alder reaction; dienes;
D O I
10.1016/S0040-4039(98)00562-0
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Synthesis of new five and seven membered outer ring diene building blocks containing alpha-amino acid moiety and their usage in the preparation of the constrained amino acid derivatives is described. (C) 1998 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码:4095 / 4098
页数:4
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