The synthesis of 2-imidazolidones on solid support by tandem aminoacylation Michael addition

被引：16

作者：

Goff, D ^{[1
]}

机构：

[1] Chiron Corp, Emeryville, CA 94608 USA

来源：

TETRAHEDRON LETTERS | 1998年 / 39卷 / 12期

关键词：

D O I：

10.1016/S0040-4039(98)00009-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Reaction of isocyanates with unsaturated amines bound to a solid support can lead either to 2-imidazolidones or 2-iminooxazolidinones depending on conditions. The imidazolidones are a useful new framework for combinatorial library synthesis. (C) 1998 Elsevier Science Ltd. All rights reserved.

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页码：1477 / 1480

页数：4

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