Diversity-oriented synthesis of fused-imidazole derivatives via Groebke-Blackburn-Bienayme reaction: a review

被引:126
作者
Devi, Nisha [1 ]
Rawal, Ravindra K. [2 ]
Singh, Virender [1 ]
机构
[1] Dr BR Ambedkar Natl Inst Technol, Dept Chem, Jalandhar 144011, Punjab, India
[2] Indo Soviet Friendship Coll Pharm, Dept Pharmaceut Chem, Moga 142001, Punjab, India
关键词
Diversity-oriented synthesis; Imidazoheterocyclic; Groebke-Blackburn-Bienayme reaction; Fused imidazole; Lewis acid; Ugi type; SOLVENT-FREE SYNTHESIS; ONE-POT SYNTHESIS; MULTICOMPONENT REACTIONS; 3-COMPONENT REACTION; IONIC LIQUIDS; ORGANIC-SYNTHESIS; COMBINATORIAL SYNTHESIS; ANNULATED PYRIDINES; BIOLOGICAL-ACTIVITY; PARALLEL SYNTHESIS;
D O I
10.1016/j.tet.2014.10.032
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
[No abstract available]
引用
收藏
页码:183 / 232
页数:50
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共 147 条
[1]   BF3/MCM-41 as nano structured solid acid catalyst for the synthesis of 3-iminoaryl-imidazo[1,2-a] pyridines [J].
Abdollahi-Alibeik, Mohammad ;
Rezaeipoor-Anari, Ali .
CATALYSIS SCIENCE & TECHNOLOGY, 2014, 4 (04) :1151-1159
[2]   Catalyst-free three-component reaction between 2-aminopyridines (or 2-aminothiazoles), aldehydes, and isocyanides in water [J].
Adib, Mehdi ;
Mahdavi, Mohammad ;
Noghani, Mahsa Alizadeh ;
Mirzaei, Peiman .
TETRAHEDRON LETTERS, 2007, 48 (41) :7263-7265
[3]   One-pot synthesis of imidazo[1,2-a]pyridines from benzyl halides or benzyl tosylates, 2-aminopyridines and isocyanides [J].
Adib, Mehdi ;
Sheikhi, Ehsan ;
Rezaei, Narjes .
TETRAHEDRON LETTERS, 2011, 52 (25) :3191-3194
[4]   Sc(OTf)3 promoted multicomponent synthesis of fluorescent imidazo[1,2-c]pyrazolo[3,4-d]pyrimidine [J].
Agrebi, Asma ;
Allouche, Fatma ;
Chabchoub, Fakher ;
El-Kaim, Laurent ;
Alves, Sergio ;
Baleizao, Carlos ;
Farinha, Jose Paulo .
TETRAHEDRON LETTERS, 2013, 54 (35) :4781-4784
[5]   An efficient synthesis of ferrocenyl imidazo[1,2-a]pyridines [J].
Akbarzadeh, Roya ;
Shakibaei, Ghazaleh Imani ;
Bazgir, Ayoob .
MONATSHEFTE FUR CHEMIE, 2010, 141 (10) :1077-1081
[6]   Synthesis of novel 5-phenylimidazo[1,2-c]quinazolin-3-amine derivatives via Groebke-Blackburn-Bienaym, multicomponent reaction [J].
Akbarzadeh, Tahmineh ;
Ebrahimi, Abolfath ;
Saeedi, Mina ;
Mahdavi, Mohammad ;
Foroumadi, Alireza ;
Shafiee, Abbas .
MONATSHEFTE FUR CHEMIE, 2014, 145 (09) :1483-1487
[7]   Scaffold oriented synthesis part 4: Design, synthesis and biological evaluation of novel 5-substituted indazoles as potent and selective kinase inhibitors employing heterocycle forming and multicomponent reactions [J].
Akritopoulou-Zanze, Irini ;
Wakefield, Brian D. ;
Gasiecki, Alan ;
Kalvin, Douglas ;
Johnson, Eric F. ;
Kovar, Peter ;
Djuric, Stevan W. .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (05) :1480-1483
[8]   Design, synthesis and in vitro antimicrobial evaluation of novel Imidazo[1,2-a]pyridine and imidazo[2,1-b][1,3]benzothiazole motifs [J].
Al-Tel, Taleb H. ;
Al-Qawasmeh, Raed A. ;
Zaarour, Rania .
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2011, 46 (05) :1874-1881
[9]   Post Groebke-Blackburn multicomponent protocol: Synthesis of new polyfunctional imidazo[1,2-a]pyridine and imidazo[1,2-a]pyrimidine derivatives as potential antimicrobial agents [J].
Al-Tel, Taleb H. ;
Al-Qawasmeh, Raed A. .
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2010, 45 (12) :5848-5855
[10]   Rapid Assembly of Polyfunctional Structures Using a One-Pot Five- and Six-Component Sequential Groebke-Blackburn/Ugi/Passerini Process [J].
Al-Tel, Taleb H. ;
Al-Qawasmeh, Raed A. ;
Voelter, Wolfgang .
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2010, 2010 (29) :5586-5593