Synthesis of 1-((5-oxo-4,5-Dihydro-1,3,4-oxadiazol-2-yl)methyl)-1H-1,2,4-triazole-3-carboxylic Acid-Application of Antibacterial activity

被引:0
作者
Brahmayya, Manuri [1 ,2 ,3 ]
Samsonu, Dasi [4 ]
Rao, Alaparthi Venkateswara [5 ]
Rao, Nelli Srinivasa [6 ]
Rao, Battula Venkateswara [1 ]
Fan, Huan-Jung [3 ]
机构
[1] Andhra Univ, Dept Engn Chem, Visakhapatnam, Andhra Pradesh, India
[2] Natl Chung Hsing Univ, Dept Chem Engn, Taichung, Taiwan
[3] HungKuang Univ, Dept Environm Engn Safety & Hlth, Taichung, Taiwan
[4] Andhra Univ, Dept Organ Chem & FDW, Visakhapatnam, Andhra Pradesh, India
[5] KL Univ, Adv Funct Mat Res Ctr, Dept Phys, Guntur, Andhra Pradesh, India
[6] Natl Chiao Tung Univ, Dept Mat Sci & Engn, Hsinchu 300, Taiwan
基金
英国科研创新办公室;
关键词
1; 2; 4-Triazole; Sodium methoxide; Hydrazine monohydrate; Hydrazide; Carbon dioxide; 3; 4-Oxadiazole; 1,3,4-OXADIAZOLES; 1,3,4-THIADIAZOLES; DERIVATIVES;
D O I
10.1007/s40010-018-0507-5
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
Synthesis of 1-((5-oxo-4,5-dihydro-1,3,4-oxadiazol-2-yl) methyl)-1H-1,2,4-triazole-3-carboxylic acid was accomplished starting with the commercially available 1,2,4-triazole-3-carboxylic acid. The conversion of hydrazide and carbon dioxide to 1,3,4-oxadiazole has been explained. Antibacterial activity also studied for some synthesized compounds.
引用
收藏
页码:621 / 627
页数:7
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