A facile one-pot three-component synthesis of benzylideneamino-3,5-dimethyl-1H-pyrazoles

被引:5
|
作者
Jilloju, Parameshwara Chary [1 ]
Vedula, Rajeswar Rao [1 ]
机构
[1] Natl Inst Technol, Dept Chem, Warangal, Telangana, India
关键词
4-Amino-5-hydrazinyl-4H-1,2,4-triazole-3-thiol; acetyl acetone; 3; 5-dimethyl-1H-pyrazole; three-component; PYRAZOLE DERIVATIVES; SCHIFF-BASES; ANTIBACTERIAL; AGENTS; TRIAZOLOTHIADIAZINES; FLUORINE;
D O I
10.1080/00397911.2018.1458242
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A facile, one-pot three-component protocol for the synthesis of substituted 4-(benzylideneamino)-5-(3,5-dimethyl-1H-pyrazol-1-yl)-4H-1,2,4-triazole-3-thiols have been reported by the reaction of 4-amino-5-hydrazinyl-4H-1,2,4-triazole-3-thiol with acetyl acetone and various substituted benzaldehydes via multi component reaction. The newly synthesized derivatives were characterized by their elemental analysis and spectral data. The current strategy provides heterocyclic compounds in good yields with broad substrate scope. [GRAPHICS] .
引用
收藏
页码:1739 / 1746
页数:8
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