An amidyl radical cyclisation approach towards the synthesis of β-lactams

被引：28
|
作者：
Clark, AJ [1 ]
Peacock, JL [1 ]
机构：
[1] Univ Warwick, Dept Chem, Coventry CV4 7AL, W Midlands, England
来源：
TETRAHEDRON LETTERS | 1998年 / 39卷 / 10期
关键词：
D O I：
10.1016/S0040-4039(97)10772-9
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Amidyl radicals generated from tributylstannane mediated homolysis of O-benzoyl hydroxamic acid derivatives (2a-d) undergo 4-exo trig cyclisation to furnish beta-lactam derivatives (4a-d). (C) 1998 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：1265 / 1268
页数：4
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