Real-time monitoring of drug release

被引:126
作者
Weinstain, Roy [1 ]
Segal, Ehud [2 ]
Satchi-Fainaro, Ronit [2 ]
Shabat, Doron [1 ]
机构
[1] Tel Aviv Univ, Raymond & Beverly Sackler Fac Exact Sci, Sch Chem, IL-69978 Tel Aviv, Israel
[2] Tel Aviv Univ, Dept Physiol & Pharmacol, Sackler Fac Med Sci, IL-69978 Tel Aviv, Israel
基金
以色列科学基金会;
关键词
TUMOR-TARGETING DEVICE; CATHEPSIN-B; DELIVERY; THERAPEUTICS; DOXORUBICIN; ANTICANCER; DENDRIMERS; CONJUGATE; PRODRUG; CELLS;
D O I
10.1039/b919329d
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
A new prodrug system, assembled using a distinctive coumarin linker, was demonstrated to report real-time activation and drug release in vitro.
引用
收藏
页码:553 / 555
页数:3
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