Structure-activity relationships of thiazole and thiadiazole derivatives as potent and selective human adenosine A3 receptor antagonists.

被引:0
|
作者
Kim, YC
Jung, KY
Kim, SK
Gao, ZG
Gross, AS
Melman, N
Jacobson, KA
机构
[1] Kwangju Inst Sci & Technol, Dept Life Sci, Kwangju 500712, South Korea
[2] NIDDK, Mol Recognit Sect, NIH, Bethesda, MD 20892 USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
255-MEDI
引用
收藏
页码:U53 / U53
页数:1
相关论文
共 50 条
  • [1] Structure-activity relationships of thiazole and thiadiazole derivatives as potent and selective human adenosine A3 receptor antagonists
    Jung, KY
    Kim, SK
    Gao, ZG
    Gross, AS
    Melman, N
    Jacobson, KA
    Kim, YC
    BIOORGANIC & MEDICINAL CHEMISTRY, 2004, 12 (03) : 613 - 623
  • [2] Structure-activity relationships of truncated adenosine derivatives as highly potent and selective human A3 adenosine receptor antagonists
    Pal, Shantanu
    Choi, Won Jun
    Choe, Seung Ah
    Heller, Cara L.
    Gao, Zhan-Guo
    Chinn, Moshe
    Jacobson, Kenneth A.
    Hou, Xiyan
    Lee, Sang Kook
    Kim, Hea Ok
    Jeong, Lak Shin
    BIOORGANIC & MEDICINAL CHEMISTRY, 2009, 17 (10) : 3733 - 3738
  • [3] Exploring 3D-QSAR of thiazole and thiadiazole derivatives as potent and selective human adenosine A3 receptor antagonists+
    Prosenjit Bhattacharya
    J. Thomas Leonard
    Kunal Roy
    Journal of Molecular Modeling, 2005, 11 : 516 - 524
  • [4] Exploring 3D-QSAR of thiazole and thiadiazole derivatives as potent and selective human adenosine A3 receptor antagonists+
    Bhattacharya, P
    Leonard, JT
    Roy, K
    JOURNAL OF MOLECULAR MODELING, 2005, 11 (06) : 516 - 524
  • [5] Exploring QSAR of thiazole and thiadiazole derivatives as potent and selective human adenosine A3 receptor antagonists using FA and GFA techniques
    Bhattacharya, P
    Leonard, JT
    Roy, K
    BIOORGANIC & MEDICINAL CHEMISTRY, 2005, 13 (04) : 1159 - 1165
  • [6] New highly potent and selective adenosine A3 receptor antagonists.
    Press, NJ
    Fozard, JR
    Beer, D
    Heng, R
    di Padova, F
    Tranter, P
    Trifilieff, A
    Walker, C
    Keller, TH
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2002, 224 : U79 - U80
  • [7] Pyrazolo Derivatives as Potent Adenosine Receptor Antagonists: An Overview on the Structure-Activity Relationships
    Cheong, Siew Lee
    Venkatesan, Gopalakrishnan
    Paira, Priyankar
    Jothibasu, Ramasamy
    Mandel, Alexander Laurence
    Federico, Stephanie
    Spalluto, Giampiero
    Pastorin, Giorgia
    INTERNATIONAL JOURNAL OF MEDICINAL CHEMISTRY, 2011, 2011
  • [8] Pyrimidine Derivatives as Potent and Selective A3 Adenosine Receptor Antagonists
    Yaziji, Vicente
    Rodriguez, David
    Gutierrez-de-Teran, Hugo
    Coelho, Alberto
    Caamano, Olga
    Garcia-Mera, Xerardo
    Brea, Jose
    Isabel Loza, Maria
    Isabel Cadavid, Maria
    Sotelo, Eddy
    JOURNAL OF MEDICINAL CHEMISTRY, 2011, 54 (02) : 457 - 471
  • [9] New potent and selective human adenosine A3 receptor antagonists
    Baraldi, PG
    Borea, PA
    TRENDS IN PHARMACOLOGICAL SCIENCES, 2000, 21 (12) : 456 - 459
  • [10] Highly potent and selective human adenosine A3 receptor antagonists: Triazoloquinazoline derivatives.
    Kim, YC
    Ji, XD
    Olah, ME
    Stiles, GL
    Jacobson, KA
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1997, 213 : 42 - MEDI