Diversity-Oriented Synthesis of Dibenzoazocines and Dibenzoazepines via a Microwave-Assisted Intramolecular A3-Coupling Reaction

被引：47
|
作者：
Bariwal, Jitender B. [1 ]
Ermolat'ev, Denis S. [1 ]
Glasnov, Toma N. [3 ]
Van Hecke, Kristof [2 ]
Mehta, Vaibhav P. [1 ]
Van Meervelt, Luc [2 ]
Kappe, C. Oliver [3 ]
Van der Eycken, Erik V. [1 ]
机构：
[1] Katholieke Univ Leuven, LOMAC, B-3001 Heverlee, Belgium
[2] Katholieke Univ Leuven, Dept Chem, B-3001 Heverlee, Belgium
[3] Karl Franzens Univ Graz, Inst Chem, Christian Doppler Lab Microwave Chem, A-8010 Graz, Austria
来源：
ORGANIC LETTERS | 2010年 / 12卷 / 12期
关键词：
BIARYL COUPLING REACTION; APOGALANTHAMINE ANALOGS; ORGANIC-SYNTHESIS; DIRECT-ADDITION; ENANTIOSELECTIVE SYNTHESIS; TERMINAL ALKYNES; SUZUKI-MIYAURA; COPPER; AMINE; (-)-STEGANACIN;
D O I：
10.1021/ol1008729
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An unprecedented, diversity-oriented strategy for the generation of 6,7-dihydro-5H-dibenzo[c,e]azepines and 5,6,7,8-tetrahydrodibenzo[c,e]azocines by a microwave-assisted copper-catalyzed intramolecular A(3)-coupling reaction is presented.
引用
收藏
页码：2774 / 2777
页数：4
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