Synthesis of new biheterocyclic compounds starting from Diazepam

被引：0

作者：

Benelbaghdadi, R

Hasnaoui, A

Lavergne, JP

机构：

[1] Fac Sci Semlalia, Lab Subst Nat & Heterocycles, Marrakech, Morocco

[2] Univ Montpellier 2, Lab Aminoacides Peptides & Prot, F-34095 Montpellier 5, France

来源：

BULLETIN DES SOCIETES CHIMIQUES BELGES | 1997年 / 106卷 / 12期

关键词：

D O I：

暂无

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

We report here a one-step synthesis of [1,2,4]triazolo[4,3-d][1,4]benzodiazepin 4, 5, and [1,2] oxazolo[5,4,b][1,4]benzodiazepine 6-8 by 1,3-dipolar cycloaddition of nitrilimines and nitrile oxides with the benzodiazepine 3.

引用

页码：813 / 815

页数：3

共 9 条

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[6] ELMESSAOUDI M, 1994, SYNTHETIC COMMUN, V24, P513
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[8] REGIOSELECTIVITY AND PERISELECTIVITY OF DIELS-ALDER REACTIONS AND 1,3-DIPOLAR CYCLO-ADDITIONS WITH A 1,2,4-TRIAZEPINE - THEORETICAL APPROACH
HASNAOUI, A
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[9] BENZODIAZEPINES .8. DIBORANE REDUCTION OF BENZODIAZEPIN-2-ONES
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