Synthesis of 2,3-Dihydroquinazoline-4(1H)-ones

被引：92

作者：

Shaterian, Hamid Reza ^{[1
]}

Oveisi, Ali Reza ^{[1
]}

Honarmand, Moones ^{[1
]}

机构：

[1] Univ Sistan & Baluchestan, Dept Chem, Fac Sci, Zahedan, Iran

来源：

SYNTHETIC COMMUNICATIONS | 2010年 / 40卷 / 08期

关键词：

Al(H2PO4)3; 3-(2'benzothiazolo)-2; 3-dihydroqunazoline-4(1H)-ones; isatoic anhydride; solvent-free; ENVIRONMENTALLY FRIENDLY PREPARATION; PERCHLORIC-ACID HCLO4-SIO2; SILICA SULFURIC-ACID; ONE-POT; AMIDOALKYL NAPHTHOLS; REUSABLE CATALYST; SOLVENT-FREE; QUINAZOLINONE DERIVATIVES; TUBULIN POLYMERIZATION; HETEROGENEOUS CATALYST;

D O I：

10.1080/00397910903064831

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient, inexpensive, and heterogeneous catalyst, [Al(H2PO4)3], was applied in a three-component, one-pot cyclocondensation reaction of isatoic anhydride with primary amines (or ammonium salts) and aldehydes to afford the corresponding quinazolinone derivatives in excellent yields. Reactions occurred under thermal solvent-free conditions. It was found that this solid acidic catalyst could be easily recovered and reused for at least three cycles without any loss of activity.

引用

页码：1231 / 1242

页数：12

共 50 条

[1] Incredible Role of Glycerol in Multicomponent Synthesis of 2,3-Dihydroquinazoline-4(1H)-ones and 1-Amidoalkyl-2-naphthols
Hajjami, Maryam
Bakhti, Fariba
Ghiasbeygi, Elahe
CROATICA CHEMICA ACTA, 2015, 88 (02) : 197 - 205
[2] Indium(III) Chloride: An Efficient Catalyst for One-pot Multicomponent Synthesis of 2,3-dihydroquinazoline-4(1H)-ones
Sahu, Adarsh
Mishra, Shweta
Sahu, Preeti
Gajbhiye, Asmita
Agrawal, Ram Kishore
CURRENT ORGANOCATALYSIS, 2018, 5 (02) : 137 - 144
[3] Citric Acid: A Green Bioorganic Catalyst for One-Pot Three-Component Synthesis of 2,3-dihydroquinazoline-4 (1H)-ones
Fahimi, Nafiseh
Sardarian, Ali Reza
CURRENT ORGANOCATALYSIS, 2016, 3 (01) : 39 - 44
[4] A Green, One-Pot Synthesis of Substituted 2,3-Dihydroquinazoline-4(1H)-ones in the Presence of N-Sulfonic Acid Pyridinium Chloride
Azimi, Seyedeh Bahareh
Azizian, Javad
SYNLETT, 2016, 27 (12) : 1836 - 1839
[5] Application of SBA-Pr-SO3H in the synthesis of 2,3-dihydroquinazoline-4(1H)-ones: characterization, UV–Vis investigations and DFT studies
Seyedeh Yasaman Afsar
Ghodsi Mohammadi Ziarani
Hoda Mollabagher
Parisa Gholamzadeh
Alireza Badiei
Ali Abolhasani Soorki
Journal of the Iranian Chemical Society, 2017, 14 : 577 - 583
[6] Application of SBA-Pr-SO3H in the synthesis of 2,3-dihydroquinazoline-4(1H)-ones: characterization, UV-Vis investigations and DFT studies
Afsar, Seyedeh Yasaman
Ziarani, Ghodsi Mohammadi
Mollabagher, Hoda
Gholamzadeh, Parisa
Badiei, Alireza
Soorki, Ali Abolhasani
JOURNAL OF THE IRANIAN CHEMICAL SOCIETY, 2017, 14 (03) : 577 - 583
[7] Efficient one-pot synthesis of 2,3-dihydroquinazoline-4(1H)-ones promoted by FeCl3/neutral Al2O3
Suo Juan Wu
Zi Qiang Zhao
Jing Shuo Gao
Bao Hua Chen
Guo Feng Chen
Research on Chemical Intermediates, 2019, 45 : 2327 - 2339
[8] Efficient one-pot synthesis of 2,3-dihydroquinazoline-4(1H)-ones promoted by FeCl3/neutral Al2O3
Wu, Suo Juan
Zhao, Zi Qiang
Gao, Jing Shuo
Chen, Bao Hua
Chen, Guo Feng
RESEARCH ON CHEMICAL INTERMEDIATES, 2019, 45 (04) : 2327 - 2339
[9] DABCO CONTAINING ACIDIC POLY( IONIC LIQUID): AN EFFICIENT CATALYST FOR THE ONE-POT PREPARATION OF 2,3-DIHYDROQUINAZOLINE-4(1H)-ONES
Mohammadi, Mohammad Kazem
Saghanezhad, Seyyed Jafar
Razzaghi-asl, Nima
BULLETIN OF THE CHEMICAL SOCIETY OF ETHIOPIA, 2017, 31 (03) : 535 - 544
[10] Ultrasonic Synthesis and Anti-phytopathogenic Fungi Activity Evaluation of 2-Sulfanylidene-2,3-dihydroquinazoline-4(1H)-one
Zhang, Jin
Cheng, Pei
Ma, Yangmin
Liu, Jia
Miao, Zhi
Fan, Chao
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2016, 36 (06) : 1368 - 1374

← 1 2 3 4 5 →