Synthesis and Antibacterial Evaluation of Benzofuran Based Di-1,2,3-triazoles

被引：10

作者：

Sunitha, V. ^{[1
]}

Kumar, A. Kishore ^{[2
]}

Shankaraiah, P. ^{[2
]}

Jalapathi, P. ^{[1
]}

Lincoln, Ch. A. ^{[3
]}

机构：

[1] Osmania Univ, Univ Coll Sci, Dept Chem, Hyderabad 500004, Telangana, India

[2] Vardhaman Coll Engn, Dept Humanities & Sci, Hyderabad 501218, Telangana, India

[3] Osmania Univ, Univ Coll Sci, Dept Chem, Hyderabad 500007, Telangana, India

来源：

RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2018年 / 88卷 / 07期

关键词：

benzofuran; 1,2,3-triazoles; click chemistry; antibacterial activity; CLICK CHEMISTRY; ANTIMICROBIAL ACTIVITY; BIOLOGICAL EVALUATION; DERIVATIVES; 1,2,3-TRIAZOLES; CYCLOADDITION;

D O I：

10.1134/S1070363218070265

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A series of novel benzofuran-1,2,3-triazole hybrid molecules are synthesized using the click chemistry approach. Structures of the synthesized compounds were assessed by IR, NMR, and mass spectroscopy. The tests of final products 10a-10l for their antibacterial activity demonstrate excellent to good activity against gram-positive and gram-negative bacteria.

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收藏

页码：1515 / 1524

页数：10

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