Suzuki coupling reaction for the solid-phase preparation of 5-substituted nicotinic acid derivatives

被引：20
作者：
Fernàndez, JC
Solé-Feu, L
Fernández-Forner, D
de la Figuera, N
Forns, P
Albericio, F
机构：
[1] Almirall Prodesfarma, Barcelona Sci Pk Unit, Barcelona 08028, Spain
[2] Almirall Prodesfarma, Res Ctr, Barcelona 08024, Spain
[3] Almirall Prodesfarma, Barcelona Biomed Res Inst, Barcelona 08028, Spain
来源：
TETRAHEDRON LETTERS | 2005年 / 46卷 / 04期
关键词：
combinatorial chemistry; Wang resin; Rink resin; Bal resin; 5-bromonicotinic acid; Suzuki coupling; solid-phase organic synthesis;
D O I：
10.1016/j.tetlet.2004.11.153
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The application of the Suzuki coupling reaction to the preparation of small combinatorial libraries using 5-bromonicotinic acid as a scaffold onto three different types of solid support (Wang, Rink, and BAL resin) is described. (C) 2004 Elsevier Ltd. All rights reserved.
引用
收藏
页码：581 / 585
页数：5
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