Study on the synthesis and biological activity of Schiff bases of 3-amino-dihydrothiophene-2-one

被引：0

作者：

Sun, Xiao-Hong ^{[1
]}

Li, Shu-Juan

Liu, Yuan-Fa

Chen, Bang

Jia, Ying-Qi

Tao, Yan

机构：

[1] Northwest Univ, Inst Chem, Xian 710069, Peoples R China

[2] NW Univ Xian, Dept Chem, Xian 710069, Peoples R China

来源：

CHINESE JOURNAL OF ORGANIC CHEMISTRY | 2007年 / 27卷 / 01期

关键词：

3-amino-dihydrothiophene-2-one; Schiff base; synthesis; biological activity;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Nine Schiff bases of 3-amino-dihydrothiophene-2-one were synthesized by reaction of substituted benzaldehyde with DL-homocysteine thiolactone hydrochloride by means of preferable reaction conditions. Seven of them were reported for the first time. The structures of the compounds were confirmed by elemental analysis, H-1 NMR and IR spectra. The biological tests showed that they were excellent biological active to several vegetable pathogen.

引用

页码：82 / 86

页数：5

共 18 条

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